SCHEMBL8091129

SCHEMBL8091129

Nc1cc(C2(S(=O)(=O)c3ccccn3)CC2)nc(-c2ccc(NC(=O)NC3CCC3)cc2)n1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 7/20 0.40
EGFR P00533 1/20 0.40
ERBB2 P04626 1/20 0.40
MET P08581 1/20 0.40
MERTK Q12866 1/20 0.40
KIT P10721 2/20 0.39
FLT3 P36888 1/20 0.39
CA12 O43570 2/20 0.39
CA1 P00915 2/20 0.39
CA2 P00918 2/20 0.39
CA9 Q16790 2/20 0.39
EPHX1 P07099 4/20 0.39
RAB9A P51151 2/20 0.39
GAA P10253 1/20 0.39
MAP4K4 O95819 1/20 0.39
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38
EPHX2 P34913 2/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
PDGFRA P16234 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8097518 0.95 KDR (0.38) KDREGFRERBB2METMERTK
SCHEMBL8090842 0.95 KDR (0.38) KDREGFRERBB2METMERTK
SCHEMBL8084833 0.88 CA12 (0.43) KDRKITFLT3CA12CA1
SCHEMBL8096070 0.87 MTOR (0.40) ATR
SCHEMBL8092294 0.86 ROCK2 (0.39) CA12CA1CA2CA9ATR
SCHEMBL8092270 0.86 NPC1 (0.43) KDRKITFLT3RAB9ASMN1; SMN2
SCHEMBL8096681 0.86 ATR (0.40) GAAATR
SCHEMBL8098135 0.85 MTOR (0.39) ATR
SCHEMBL8099411 0.84 CA12 (0.44) KDRKITFLT3CA12CA1
SCHEMBL8091924 0.83 NAMPT (0.39) KDRKITCA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed