SCHEMBL8099563

SCHEMBL8099563

Cc1nc(C)c(S(=O)(=O)C2(c3cc(N)nc(-c4ccc(NC(=O)NCCF)cc4)n3)CC2)s1

nearest known ligand 0.38

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
PIK3CA P42336 12/20 0.38
MTOR P42345 11/20 0.38
PIK3CD O00329 6/20 0.37
KDM4E B2RXH2 2/20 0.35
RAB9A P51151 2/20 0.35
GAA P10253 1/20 0.35
SMN1; SMN2 Q16637 2/20 0.34
NPC1 O15118 1/20 0.34
GLA P06280 1/20 0.34
ALDH1A1 P00352 1/20 0.33
POLB P06746 1/20 0.33
PIK3CG P48736 2/20 0.33
ATR Q13535 1/20 0.33
PIK3CB P42338 1/20 0.33
KIT P10721 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8098739 0.90 PIK3CD (0.36) PIK3CAMTORPIK3CDKDM4ERAB9A
SCHEMBL8107169 0.88 MTOR (0.37) PIK3CAMTORPIK3CDPIK3CGKIT
SCHEMBL8099632 0.85 CA1 (0.42) PIK3CAMTORPIK3CDRAB9AALDH1A1
SCHEMBL8091538 0.84 PIK3CD (0.43) PIK3CAMTORPIK3CDPIK3CGATR
SCHEMBL8084009 0.84 PIK3CD (0.42) PIK3CAMTORPIK3CDPIK3CGATR
SCHEMBL8104327 0.84 NAMPT (0.39) PIK3CAMTORPIK3CD
SCHEMBL8091534 0.83 NAMPT (0.40) PIK3CAMTORPIK3CDSMN1; SMN2ALDH1A1
SCHEMBL8091717 0.83 CA2 (0.40) PIK3CAMTORPIK3CDKDM4E
SCHEMBL8107163 0.82 KDM4E (0.42) PIK3CAMTORPIK3CDKDM4ERAB9A
SCHEMBL8100136 0.82 NAMPT (0.41) PIK3CAMTORPIK3CDKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed