SCHEMBL8100175

SCHEMBL8100175

O=c1cc(-c2cccc(Cl)c2)nc2ccccn12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRM5 P41594 1/20 0.55
KDM5B Q9UGL1 1/20 0.51
KDM4E B2RXH2 4/20 0.46
ALDH1A1 P00352 3/20 0.46
POLB P06746 2/20 0.46
GAA P10253 2/20 0.46
HPGD P15428 2/20 0.46
GLA P06280 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HSD17B10 Q99714 1/20 0.46
NPC1 O15118 1/20 0.44
RAB9A P51151 1/20 0.44
MAPT P10636 5/20 0.44
KMT2A Q03164 3/20 0.44
LMNA P02545 2/20 0.44
PSD A5PKW4 1/20 0.44
ADORA3 P0DMS8 1/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
ADORA1 P30542 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8105987 0.85 NPC1 (0.55) GRM5KDM5BKDM4EALDH1A1POLB
SCHEMBL1659994 0.85 KDM4E (0.52) GRM5KDM5BKDM4EALDH1A1GAA
SCHEMBL31365868 0.83 KDM5B (0.50) GRM5KDM5BKDM4EALDH1A1POLB
SCHEMBL28958139 0.83 KDM5B (0.50) GRM5KDM5BKDM4EALDH1A1POLB
SCHEMBL8105559 0.83 RAB9A (0.54) KDM4EALDH1A1POLBGAAHPGD
SCHEMBL8102024 0.82 ALDH1A1 (0.55) KDM5BKDM4EALDH1A1POLBNPC1
SCHEMBL7925220 0.80 MEN1 (0.57) KDM4EALDH1A1HPGDHSD17B10NPC1
SCHEMBL8102158 0.80 NR1H4 (0.50) KDM5BKDM4EALDH1A1HPGDHSD17B10
SCHEMBL8099804 0.79 RAB9A (0.49) GRM5KDM4EALDH1A1GAAHPGD
SCHEMBL1659969 0.79 NPC1 (0.47) KDM5BKDM4EALDH1A1HPGDNPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6071930-A FOR INHIBITION OF MITOSIS OR TUMOR GROWTH THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 2000-06-06 US disclosed
US-5994367-A PREVENT CELL MITOSIS; ANTICARCINOGENIC AGENTS THE UNIVERSITY OF NORTH CAROLINA AT CHAPEL HILL (US) 1999-11-30 US disclosed