SCHEMBL28958139

SCHEMBL28958139

O=c1cc(-c2cccc(F)c2)nc2ccccn12

nearest known ligand 0.63

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM5B Q9UGL1 1/20 0.50
KMT2A Q03164 3/20 0.46
CDC7 O00311 1/20 0.46
PIM1 P11309 1/20 0.46
GSK3B P49841 1/20 0.46
HIPK2 Q9H2X6 1/20 0.46
CLK4 Q9HAZ1 1/20 0.46
MAPT P10636 4/20 0.43
TP53 P04637 1/20 0.43
THRB P10828 1/20 0.43
KDM4E B2RXH2 5/20 0.43
ADORA3 P0DMS8 2/20 0.43
ADORA2A P29274 1/20 0.43
ADORA2B P29275 1/20 0.43
ADORA1 P30542 1/20 0.43
PRKDC P78527 1/20 0.43
HPGD P15428 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MAOB P27338 1/20 0.42
ALDH1A1 P00352 3/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31365868 1.00 KDM5B (0.50) KDM5BKMT2ACDC7PIM1GSK3B
SCHEMBL8092386 0.85 NPC1 (0.55) KDM5BKMT2ACDC7PIM1GSK3B
SCHEMBL1659994 0.85 KDM4E (0.52) KDM5BKMT2AMAPTTP53THRB
SCHEMBL8100175 0.83 GRM5 (0.55) KDM5BKMT2APIM1GSK3BHIPK2
SCHEMBL8105559 0.83 RAB9A (0.54) KMT2AMAPTKDM4EADORA3ADORA2A
SCHEMBL7925220 0.80 MEN1 (0.57) KMT2AMAPTTP53KDM4EADORA3
SCHEMBL8100231 0.80 GRIN1 (0.49) KDM5BKMT2ACDC7PIM1GSK3B
SCHEMBL8099804 0.79 RAB9A (0.49) KMT2AMAPTKDM4EADORA3ADORA2A
SCHEMBL1834856 0.78 ADORA3 (0.47) KDM5BKMT2ACDC7PIM1GSK3B
SCHEMBL8105987 0.77 NPC1 (0.55) KDM5BKMT2AMAPTKDM4EADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115557948-A Method for preparing pyrido [1,2-a ] pyrimidin-4-one compound selenized at C3 position 淄博职业学院 2023-01-03 CN claimed
CN-115557948-A Method for preparing pyrido [1,2-a ] pyrimidin-4-one compound selenized at C3 position 淄博职业学院 2023-01-03 CN disclosed