SCHEMBL8101941

SCHEMBL8101941

Cc1cc(CC2CCN(Cc3cccnc3)CC2)c2cccc(F)c2n1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.45
ALDH1A1 P00352 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
TRPV6 Q9H1D0 1/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
KMT2A Q03164 2/20 0.42
MEN1 O00255 1/20 0.42
NPC1 O15118 1/20 0.42
MAPT P10636 1/20 0.42
BLM P54132 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
ATM Q13315 1/20 0.42
TSHR P16473 2/20 0.41
LMNA P02545 1/20 0.41
CACNA1I Q9P0X4 1/20 0.41
PDE2A O00408 1/20 0.41
HTR1A P08908 2/20 0.41
HTR1D P28221 1/20 0.41
HTR1B P28222 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13945322 0.83 SCN9A (0.46) KDM4EALDH1A1TDP1TRPV6CHRNB2
SCHEMBL8095854 0.79 KDM4E (0.46) KDM4EALDH1A1TDP1KMT2AMEN1
SCHEMBL8102177 0.78 GPR6 (0.47) KDM4EALDH1A1KMT2AMEN1ATM
SCHEMBL8092993 0.78 HTR2B (0.44) ATMHTR1AHTR2CHTR7HTR2B
SCHEMBL21063255 0.77 ADORA2A (0.45) KDM4EALDH1A1TDP1CHRNB2CHRNA4
SCHEMBL8102227 0.75 GRIN1 (0.42) KDM4EKMT2AMEN1NPC1MAPT
SCHEMBL8100325 0.71 JAK2 (0.39) ALDH1A1NPC1HTR1AHTR2CHTR7
SCHEMBL5526683 0.71 SCN1A (0.50) KDM4ESMN1; SMN2
SCHEMBL8430036 0.71 CHRNB2 (0.64) KDM4EALDH1A1TDP1TRPV6CHRNB2
SCHEMBL803669 0.69 CHRNB2 (0.60) KDM4EALDH1A1TDP1TRPV6CHRNB2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000085-A1 QUINOLINE AND QUINAZOLINE DERIVATIVES USEFUL AS MODULATORS OF GATED ION CHANNELS PAINCEPTOR PHARMA CORPORATION (CA) 2008-12-31 WO disclosed