SCHEMBL8102227

SCHEMBL8102227

CNC(=N)c1ccccc1CN1CCC(Cc2cc(C)nc3c(F)cccc23)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRIN1 Q05586 2/20 0.42
GRIN2B Q13224 2/20 0.42
ATM Q13315 1/20 0.41
KMT2A Q03164 3/20 0.41
MEN1 O00255 2/20 0.41
DRD4 P21917 1/20 0.40
CCR3 P51677 3/20 0.40
DRD2 P14416 1/20 0.40
HTR2A P28223 1/20 0.40
HRH1 P35367 1/20 0.40
ACHE P22303 1/20 0.38
HTR2C P28335 1/20 0.38
HTR7 P34969 1/20 0.38
HTR2B P41595 1/20 0.38
HTR3A P46098 1/20 0.38
HTR4 Q13639 1/20 0.38
KDM4E B2RXH2 1/20 0.38
NPC1 O15118 1/20 0.38
MAPT P10636 1/20 0.38
BLM P54132 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8092993 0.80 HTR2B (0.44) GRIN1GRIN2BATMCCR3DRD2
SCHEMBL8095854 0.77 KDM4E (0.46) GRIN1GRIN2BATMKMT2AMEN1
SCHEMBL8097090 0.76 DRD4 (0.37) KMT2AMEN1DRD4ACHEPHGDH
SCHEMBL8102177 0.76 GPR6 (0.47) ATMKMT2AMEN1KDM4ESLC6A4
SCHEMBL8101941 0.75 KDM4E (0.45) ATMKMT2AMEN1HTR2CHTR7
SCHEMBL8095852 0.72 CCR3 (0.47) GRIN1GRIN2BATMKMT2AMEN1
SCHEMBL8091662 0.71 HRH1 (0.47) KMT2ADRD4CCR3HRH1
SCHEMBL8095680 0.69 PDE4B (0.46) ATMKMT2AMEN1ACHEHTR2C
SCHEMBL13945410 0.67 MEN1 (0.39) ATMKMT2AMEN1DRD4CCR3
SCHEMBL13968360 0.66 OPRL1 (0.42) KMT2AMEN1DRD4CCR3HRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009000085-A1 QUINOLINE AND QUINAZOLINE DERIVATIVES USEFUL AS MODULATORS OF GATED ION CHANNELS PAINCEPTOR PHARMA CORPORATION (CA) 2008-12-31 WO disclosed