SCHEMBL8102565

SCHEMBL8102565

CCCCN1CCN(N2C(=O)c3ccccc3C2=O)CC1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.50
HTR1A P08908 5/20 0.48
DRD2 P14416 2/20 0.47
CHRM2 P08172 1/20 0.47
CHRM4 P08173 1/20 0.47
CHRM5 P08912 1/20 0.47
CHRM1 P11229 1/20 0.47
CHRM3 P20309 1/20 0.47
DRD4 P21917 1/20 0.47
DRD3 P35462 1/20 0.47
HTR2A P28223 1/20 0.45
HTR6 P50406 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7083799 0.95 MAOB (0.52) MAOBHTR1ADRD2DRD3
SCHEMBL8092753 0.90 DRD2 (0.49) MAOBHTR1ADRD2
SCHEMBL6953084 0.83 MAOB (0.62) MAOBHTR1A
SCHEMBL6946848 0.83 MAOB (0.71) MAOBHTR1ADRD2DRD3
Hydrochloric Acid SCHEMBL31491133 0.81 HTR1A (0.48) MAOBHTR1ACHRM2CHRM4CHRM5
SCHEMBL30022123 0.79 POLB (0.54)
Hydrochloric Acid SCHEMBL31491177 0.77 SIGMAR1 (0.43) MAOBHTR1ACHRM2CHRM4CHRM5
SCHEMBL5232218 0.74 ACHE (0.52) MAOBHTR1ADRD2CHRM2CHRM4
SCHEMBL14028451 0.73 HTR1A (0.79) MAOBHTR1ADRD2DRD3
SCHEMBL13469510 0.73 HTR1A (0.79) MAOBHTR1ADRD2DRD3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130030007-A1 Obesity Small Molecules AKRON MOLECULES GMBH (AT) 2013-01-31 US disclosed
US-6057371-A TREATMENT OF CENTRAL NERVOUS SYSTEM DISORDERS, GASTROINTESTINAL DISORDERS, DRUG ABUSE, ANGINA, MIGRAINE, HYPERTENSION AND DEPRESSION VIRGINIA COMMONWEALTH UNIVERSITY (US) 2000-05-02 US disclosed