SCHEMBL8103655

SCHEMBL8103655

CCCCc1ccc(C(=O)Cl)cc1.CCCc1ccc(C(=O)Cl)cc1

nearest known ligand 0.59

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
RARB P10826 6/20 0.59
PLK1 P53350 2/20 0.59
THRB P10828 6/20 0.57
THRA P10827 5/20 0.57
ALDH1A1 P00352 3/20 0.55
HPGD P15428 1/20 0.55
HSD17B10 Q99714 1/20 0.55
KDM4E B2RXH2 1/20 0.51
POLB P06746 1/20 0.51
GAA P10253 1/20 0.51
CTDSP1 Q9GZU7 1/20 0.51
MEN1 O00255 1/20 0.51
RARA P10276 1/20 0.51
MAPT P10636 1/20 0.51
MTOR P42345 1/20 0.51
KMT2A Q03164 1/20 0.51
TRPV1 Q8NER1 1/20 0.51
L3MBTL1 Q9Y468 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1020423 0.96 RARB (0.62) RARBPLK1THRBTHRAALDH1A1
SCHEMBL1019681 0.92 PLK1 (0.60) RARBPLK1THRBTHRAALDH1A1
SCHEMBL12656104 0.91 RARB (0.72) RARBPLK1THRBTHRAALDH1A1
SCHEMBL158152 0.91 THRA (0.67) RARBTHRBTHRAALDH1A1MEN1
SCHEMBL7728431 0.91 THRA (0.59) RARBTHRBTHRAALDH1A1MEN1
SCHEMBL1020543 0.89 THRA (0.70) RARBTHRBTHRAALDH1A1MEN1
SCHEMBL8960387 0.89 THRA (0.70) RARBTHRBTHRAALDH1A1MEN1
SCHEMBL17272985 0.89 THRA (0.70) RARBTHRBTHRAALDH1A1MEN1
SCHEMBL8728345 0.89 THRA (0.70) RARBTHRBTHRAALDH1A1MEN1
SCHEMBL2180222 0.89 THRA (0.70) RARBTHRBTHRAALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed