SCHEMBL8103978

SCHEMBL8103978

CNC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)O)CC3)n2)cn1

nearest known ligand 0.37

Predicted protein targets (top 4)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 3/20 0.37
MAP4K1 Q92918 4/20 0.36
GCK P35557 3/20 0.32
APP P05067 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099234 0.89 KCNH2 (0.35) ABL1APP
SCHEMBL8098261 0.86 MTOR (0.43)
SCHEMBL8092878 0.79 NPC1 (0.46)
SCHEMBL8092946 0.76 ABL1 (0.41) ABL1
SCHEMBL8095600 0.76 CA12 (0.39) MAP4K1
SCHEMBL8090594 0.74 PIK3CD (0.40)
SCHEMBL8092884 0.73 KDR (0.41)
SCHEMBL8089827 0.73 PIK3CD (0.37)
SCHEMBL8213772 0.72 PIK3CD (0.38) ABL1MAP4K1
SCHEMBL8083714 0.72 EPHX1 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed