SCHEMBL8092946

SCHEMBL8092946

CNC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccc(F)cc4)CC3)n2)cn1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 2/20 0.41
PIK3R1 P27986 1/20 0.38
PIK3CA P42336 1/20 0.38
NPC1 O15118 1/20 0.35
RAB9A P51151 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
ALDH1A1 P00352 1/20 0.35
TDO2 P48775 3/20 0.35
DGAT1 O75907 2/20 0.35
RORC P51449 4/20 0.34
KDR P35968 1/20 0.34
TEK Q02763 1/20 0.34
CA12 O43570 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34
CA9 Q16790 1/20 0.34
PSEN1 P49768 2/20 0.33
PSEN2 P49810 2/20 0.33
APH1B Q8WW43 2/20 0.33
NCSTN Q92542 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099954 0.89 ABL1 (0.40) ABL1PIK3R1PIK3CASMN1; SMN2RORC
SCHEMBL8083973 0.88 ALDH1A1 (0.43) PIK3R1PIK3CANPC1RAB9AALDH1A1
SCHEMBL8083683 0.81 NPC1 (0.42) PIK3R1PIK3CANPC1RAB9ASMN1; SMN2
SCHEMBL8089917 0.81 PIK3CA (0.39) PIK3CAALDH1A1CA2CA9NAMPT
SCHEMBL8092637 0.81 KMT2A (0.42) PIK3CACA12CA1CA2CA9
SCHEMBL3926957 0.80 PIK3CA (0.47) PIK3R1PIK3CA
SCHEMBL8083334 0.80 CA1 (0.41) PIK3R1PIK3CAALDH1A1CA12CA1
SCHEMBL8097257 0.80 ALDH1A1 (0.41) PIK3CARAB9AALDH1A1CA12CA1
SCHEMBL8094619 0.80 PIP4K2A (0.40) PIK3R1PIK3CANAMPT
SCHEMBL8083200 0.79 ALDH1A1 (0.43) PIK3R1PIK3CAALDH1A1TDO2CA12

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed