SCHEMBL8104255

SCHEMBL8104255

Fc1ccccc1-c1[c]c[nH]n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOTUM Q6P988 2/20 0.42
IDO1 P14902 1/20 0.42
DCUN1D1 Q96GG9 2/20 0.39
NISCH Q9Y2I1 1/20 0.37
ALDH1A1 P00352 3/20 0.36
NPC1 O15118 2/20 0.36
PKM P14618 1/20 0.36
RAB9A P51151 1/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
KDM4E B2RXH2 1/20 0.34
HTR7 P34969 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CCNE2 O96020 1/20 0.34
CCNE1 P24864 1/20 0.34
CDK2 P24941 1/20 0.34
TNKS O95271 1/20 0.33
TNKS2 Q9H2K2 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ALOX15 P16050 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6623237 0.77 ALDH1A1 (0.42) NOTUMIDO1DCUN1D1NISCHALDH1A1
SCHEMBL9903469 0.77 NOTUM (0.46) NOTUM
SCHEMBL7853517 0.70 NOTUM (0.45) NOTUMIDO1
SCHEMBL4630228 0.70 IDO1 (0.33) IDO1ALDH1A1NPC1L3MBTL1KDM4E
SCHEMBL28018833 0.65 KDM4E (0.39) NOTUMIDO1DCUN1D1NISCHALDH1A1
SCHEMBL29547174 0.65 ACHE (0.47) NOTUMIDO1DCUN1D1NISCHALDH1A1
SCHEMBL197834 0.65 ACHE (0.47) NOTUMIDO1DCUN1D1NISCHALDH1A1
SCHEMBL8117022 0.65 NFE2L2 (0.53) NPC1PKMRAB9AL3MBTL1KDM4E
SCHEMBL30497931 0.64 IDO1 (0.53) NOTUMIDO1DCUN1D1NISCHALDH1A1
SCHEMBL2277157 0.64 IDO1 (0.53) NOTUMIDO1DCUN1D1NISCHALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1000055-A1 SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS G.D. Searle & Co. (US) 2000-05-17 EP disclosed
WO-1998052940-A1 SUBSTITUTED PYRAZOLES AS p38 KINASE INHIBITORS G.D. SEARLE AND CO. (US) 1998-11-26 WO disclosed