SCHEMBL4630228

SCHEMBL4630228

Nc1cccc(-c2[c]c[nH]n2)c1N

nearest known ligand 0.33

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.33
CD44 P16070 1/20 0.32
ALDH1A1 P00352 2/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KDM4E B2RXH2 2/20 0.31
NPC1 O15118 1/20 0.31
GAA P10253 1/20 0.31
HSD17B10 Q99714 1/20 0.31
PPARG P37231 1/20 0.30
NCOA2 Q15596 1/20 0.30
NCOA1 Q15788 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30
NPSR1 Q6W5P4 1/20 0.30
RXFP1 Q9HBX9 1/20 0.30
TDP1 Q9NUW8 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104255 0.70 NOTUM (0.42) IDO1ALDH1A1L3MBTL1KDM4ENPC1
SCHEMBL6623237 0.70 ALDH1A1 (0.42) IDO1ALDH1A1L3MBTL1KDM4ENPC1
SCHEMBL560128 0.68 ALDH1A1 (0.56) CD44ALDH1A1L3MBTL1HSD17B10SMN1; SMN2
SCHEMBL5236188 0.67 IDO1 (0.38) IDO1CD44ALDH1A1L3MBTL1KDM4E
Hydrochloric Acid SCHEMBL4521251 0.66 ALDH1A1 (0.53) CD44ALDH1A1L3MBTL1HSD17B10SMN1; SMN2
Methane SCHEMBL22720568 0.66 ALDH1A1 (0.53) CD44ALDH1A1L3MBTL1HSD17B10SMN1; SMN2
SCHEMBL28448451 0.64 ALDH1A1 (0.58) CD44ALDH1A1L3MBTL1HSD17B10SMN1; SMN2
SCHEMBL169282 0.63 ALDH1A1 (0.68) CD44ALDH1A1L3MBTL1KDM4ENPC1
SCHEMBL29564016 0.63 ALDH1A1 (0.68) CD44ALDH1A1L3MBTL1KDM4ENPC1
SCHEMBL15364728 0.63 IMPDH2 (0.51) CD44ALDH1A1L3MBTL1NPC1HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1919907-A2 HETEROCYCLIC COMPOUND OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2008-05-14 EP disclosed
WO-2007026959-A2 DERIVATIVES OF 4-PIPERAZIN-1-YL-4-BENZ0 [B] THIOPHENE SUITABLE FOR THE TREATMENT OF CNS DISORDERS OTSUKA PHARMACEUTICAL CO., LTD. (JP) 2007-03-08 WO disclosed