SCHEMBL8104401

SCHEMBL8104401

CC(C)Oc1ccc(NC(=O)CN(Cc2cn(C(=O)OC(C)(C)C)cn2)c2cccc(C#N)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 1/20 0.38
PSMB5 P28074 2/20 0.37
ALDH1A1 P00352 4/20 0.36
MAPT P10636 3/20 0.36
LMNA P02545 2/20 0.36
MAPK1 P28482 1/20 0.36
HTT P42858 1/20 0.34
RORC P51449 2/20 0.34
KIT P10721 1/20 0.34
CETP P11597 1/20 0.33
TP53 P04637 1/20 0.33
POLB P06746 1/20 0.33
KMT2A Q03164 1/20 0.33
NLRP1 Q9C000 1/20 0.33
GCK P35557 1/20 0.32
ABL1 P00519 1/20 0.32
KCNH2 Q12809 1/20 0.32
PFKFB2 O60825 1/20 0.32
PFKFB1 P16118 1/20 0.32
PFKFB3 Q16875 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104036 0.91 MCHR1 (0.38) MCHR1PSMB5ALDH1A1MAPTLMNA
SCHEMBL8120737 0.82 MAOB (0.35)
SCHEMBL8112927 0.79 MCHR1 (0.37) MCHR1PSMB5ALDH1A1MAPTHTT
SCHEMBL8113921 0.78 RORC (0.46) MCHR1PSMB5ALDH1A1MAPTLMNA
SCHEMBL8112799 0.78 PSMB5 (0.47) MCHR1PSMB5ALDH1A1MAPTLMNA
SCHEMBL8113481 0.77 RORC (0.37) MCHR1PSMB5ALDH1A1MAPTLMNA
SCHEMBL8104607 0.77 RORC (0.36) ALDH1A1LMNAHTTRORCKMT2A
SCHEMBL8113210 0.76 ALDH1A1 (0.41) MCHR1PSMB5ALDH1A1MAPTLMNA
SCHEMBL8104603 0.76 MCHR1 (0.46) MCHR1PSMB5ALDH1A1MAPTLMNA
SCHEMBL8119058 0.75 MCHR1 (0.45) MCHR1PSMB5ALDH1A1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020434-A1 3-AMIDINOANILINE DERIVATIVES, ACTIVATED BLOOD COAGULATION FACTOR X INHIBITORS, AND INTERMEDIATES FOR PRODUCING BOTH Kissei Pharmaceutical Co., Ltd. (JP) 2000-07-19 EP disclosed