SCHEMBL8104036

SCHEMBL8104036

CC(C)c1ccc(NC(=O)CN(Cc2cn(C(=O)OC(C)(C)C)cn2)c2cccc(C#N)c2)cc1

nearest known ligand 0.38

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 3/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPT P10636 2/20 0.37
PANK3 Q9H999 2/20 0.36
HTT P42858 1/20 0.35
NPC1 O15118 2/20 0.35
RAB9A P51151 2/20 0.35
PSMB5 P28074 1/20 0.35
RORC P51449 2/20 0.34
LMNA P02545 2/20 0.34
TP53 P04637 1/20 0.34
MAPK1 P28482 1/20 0.34
SMN1; SMN2 Q16637 1/20 0.33
CETP P11597 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104401 0.91 MCHR1 (0.38) MCHR1ALDH1A1MAPTHTTPSMB5
SCHEMBL8112927 0.88 MCHR1 (0.37) MCHR1ALDH1A1MAPTPANK3HTT
SCHEMBL8113481 0.86 RORC (0.37) MCHR1ALDH1A1MAPTPANK3HTT
SCHEMBL8113210 0.86 ALDH1A1 (0.41) MCHR1ALDH1A1MAPTPANK3HTT
SCHEMBL8120737 0.84 MAOB (0.35)
SCHEMBL8118821 0.83 ALDH1A1 (0.40) MCHR1ALDH1A1MAPTPANK3HTT
SCHEMBL8112410 0.80 NLRP3 (0.38) MCHR1ALDH1A1MAPTPANK3HTT
SCHEMBL8104244 0.80 THRB (0.40) MCHR1ALDH1A1MAPTPANK3HTT
SCHEMBL8113521 0.78 MAPT (0.42) MCHR1ALDH1A1MAPTPANK3HTT
SCHEMBL8104607 0.78 RORC (0.36) ALDH1A1HTTRORCLMNASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020434-A1 3-AMIDINOANILINE DERIVATIVES, ACTIVATED BLOOD COAGULATION FACTOR X INHIBITORS, AND INTERMEDIATES FOR PRODUCING BOTH Kissei Pharmaceutical Co., Ltd. (JP) 2000-07-19 EP disclosed