SCHEMBL8112927

SCHEMBL8112927

CC(C)c1ccc(NC(=O)CN(Cc2cn(CC(=O)OC(C)(C)C)cn2)c2cccc(C#N)c2)cc1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 3/20 0.37
ALDH1A1 P00352 3/20 0.36
MAPT P10636 2/20 0.36
GAA P10253 1/20 0.36
POLB P06746 1/20 0.36
PANK3 Q9H999 1/20 0.35
TP53 P04637 1/20 0.34
HTT P42858 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
PSMB5 P28074 1/20 0.34
KMT2A Q03164 1/20 0.34
RORC P51449 1/20 0.34
FNTA P49354 2/20 0.33
FNTB P49356 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104036 0.88 MCHR1 (0.38) MCHR1ALDH1A1MAPTPANK3TP53
SCHEMBL8118821 0.87 ALDH1A1 (0.40) MCHR1ALDH1A1MAPTGAAPOLB
SCHEMBL8113210 0.84 ALDH1A1 (0.41) MCHR1ALDH1A1MAPTPOLBPANK3
SCHEMBL8104244 0.84 THRB (0.40) MCHR1ALDH1A1MAPTPOLBPANK3
SCHEMBL8112410 0.84 NLRP3 (0.38) MCHR1ALDH1A1MAPTGAAPOLB
SCHEMBL8113481 0.81 RORC (0.37) MCHR1ALDH1A1MAPTPANK3TP53
SCHEMBL8104401 0.79 MCHR1 (0.38) MCHR1ALDH1A1MAPTPOLBTP53
Hydrochloric Acid SCHEMBL8118540 0.78 F10 (0.43) ALDH1A1MAPTPOLBTP53RAB9A
SCHEMBL8113521 0.77 MAPT (0.42) MCHR1ALDH1A1MAPTPOLBPANK3
SCHEMBL27538508 0.76 LMNA (0.54) MCHR1ALDH1A1MAPTPOLBHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1268116-A 3-amidinoaniline derivatives activated blood coagulation factor X inhibitors, and intermediates for producing both KISSEI PHARMACEUTICAL (JP) 2000-09-27 CN disclosed
EP-1020434-A1 3-AMIDINOANILINE DERIVATIVES, ACTIVATED BLOOD COAGULATION FACTOR X INHIBITORS, AND INTERMEDIATES FOR PRODUCING BOTH Kissei Pharmaceutical Co., Ltd. (JP) 2000-07-19 EP disclosed