SCHEMBL8104718

SCHEMBL8104718

CCCC(c1c[nH]cn1)N(CC(=O)O)c1cccc(C#N)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNN4 O15554 1/20 0.37
KCNA5 P22460 1/20 0.37
MAOB P27338 1/20 0.36
S1PR1 P21453 2/20 0.34
MMP12 P39900 1/20 0.34
MMP13 P45452 1/20 0.34
FFAR1 O14842 3/20 0.33
FFAR4 Q5NUL3 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.33
GRM5 P41594 1/20 0.32
LRRK2 Q5S007 1/20 0.32
SLC6A2 P23975 1/20 0.31
SLC6A4 P31645 1/20 0.31
SLC6A3 Q01959 1/20 0.31
GRK6 P43250 1/20 0.31
PIN1 Q13526 1/20 0.31
FOLH1 Q04609 1/20 0.31
KDM4C Q9H3R0 1/20 0.31
PER2 O15055 1/20 0.31
CRY1 Q16526 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104713 0.86 MAOB (0.40) KCNN4KCNA5MAOBS1PR1MMP12
SCHEMBL8118826 0.84 MAPT (0.38)
SCHEMBL8120742 0.79 MAOB (0.36) KCNN4KCNA5MAOBFFAR1FFAR4
SCHEMBL8112413 0.71 NLRP3 (0.36) MAOB
SCHEMBL8113212 0.70 MAPT (0.38)
SCHEMBL6979204 0.69 MAOB (0.46) KCNN4KCNA5MAOBS1PR1MMP12
SCHEMBL8104610 0.69 POLB (0.35) MAOBFFAR1FFAR4
SCHEMBL6982499 0.68 KCNN4 (0.54) KCNN4KCNA5MAOBMMP12MMP13
SCHEMBL3830265 0.67 KCNN4 (0.47) KCNN4KCNA5MAOBMMP12MMP13
SCHEMBL7057421 0.67 FFAR1 (0.47) KCNN4KCNA5MAOBMMP12MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1268116-A 3-amidinoaniline derivatives activated blood coagulation factor X inhibitors, and intermediates for producing both KISSEI PHARMACEUTICAL (JP) 2000-09-27 CN disclosed
EP-1020434-A1 3-AMIDINOANILINE DERIVATIVES, ACTIVATED BLOOD COAGULATION FACTOR X INHIBITORS, AND INTERMEDIATES FOR PRODUCING BOTH Kissei Pharmaceutical Co., Ltd. (JP) 2000-07-19 EP disclosed