SCHEMBL8112413

SCHEMBL8112413

CC(C)c1ccc(NC(=O)CN(c2cccc(C#N)c2)C(Cc2ccc(O)cc2)c2c[nH]cn2)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NLRP3 Q96P20 1/20 0.36
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.36
PSMB5 P28074 1/20 0.35
MAOB P27338 1/20 0.34
POLB P06746 1/20 0.34
CNR1 P21554 3/20 0.34
CNR2 P34972 2/20 0.34
PANK3 Q9H999 1/20 0.34
RAB9A P51151 2/20 0.34
LMNA P02545 1/20 0.34
HTT P42858 1/20 0.34
GAA P10253 1/20 0.33
CRHBP P24387 1/20 0.33
CRHR2 Q13324 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
NPC1 O15118 1/20 0.33
MCHR1 Q99705 3/20 0.33
MAP2K2 P36507 1/20 0.32
CALCRL Q16602 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8104245 0.94 RORC (0.38) MAPTALDH1A1PSMB5POLBCNR1
SCHEMBL8118826 0.88 MAPT (0.38) MAPTALDH1A1PSMB5PANK3RAB9A
SCHEMBL8113212 0.86 MAPT (0.38) MAPTALDH1A1PSMB5PANK3RAB9A
Hydrochloric Acid SCHEMBL8118843 0.85 NLRP3 (0.35) NLRP3MAPTLMNAGAACRHBP
SCHEMBL8112930 0.84 ALDH1A1 (0.35) MAPTALDH1A1PSMB5PANK3RAB9A
SCHEMBL8104039 0.80 RAB9A (0.35) MAPTALDH1A1PSMB5PANK3RAB9A
SCHEMBL8113521 0.77 MAPT (0.42) MAPTALDH1A1PSMB5POLBPANK3
Hydrochloric Acid SCHEMBL8104643 0.73 ITGB3 (0.34) MAPTRAB9ALMNASMN1; SMN2NPC1
SCHEMBL8113537 0.72 ALDH1A1 (0.48) MAPTALDH1A1POLBCNR1RAB9A
Hydrochloric Acid SCHEMBL8118543 0.71 F2 (0.37) RAB9ASMN1; SMN2NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020434-A1 3-AMIDINOANILINE DERIVATIVES, ACTIVATED BLOOD COAGULATION FACTOR X INHIBITORS, AND INTERMEDIATES FOR PRODUCING BOTH Kissei Pharmaceutical Co., Ltd. (JP) 2000-07-19 EP disclosed