SCHEMBL8106435

SCHEMBL8106435

Cn1nc(Cl)n(-c2cccc3ccc(O)cc23)c1=O

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
HTR5A P47898 1/20 0.43
MCL1 Q07820 1/20 0.39
TDP1 Q9NUW8 1/20 0.38
GSK3A P49840 1/20 0.38
GSK3B P49841 1/20 0.38
TRPV1 Q8NER1 10/20 0.38
CYP17A1 P05093 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
MTNR1A P48039 1/20 0.35
MTNR1B P49286 1/20 0.35
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8100124 0.82 SMN1; SMN2 (0.45) HTR5ACYP17A1CYP3A4CYP11B1CYP11B2
SCHEMBL8100298 0.82 HTR5A (0.41) HTR5AMCL1TDP1GSK3AGSK3B
SCHEMBL7061200 0.70 HTR5A (0.47) HTR5AMCL1TDP1TRPV1
SCHEMBL6603431 0.69 HCAR1 (0.48) TDP1
SCHEMBL28760463 0.68 HTR5A (0.51) HTR5AMCL1TDP1TRPV1ESR1
SCHEMBL13330266 0.67 MEN1 (0.54) HTR5AMCL1TRPV1CYP17A1CYP3A4
SCHEMBL6306922 0.66 HTR5A (0.68) HTR5AMCL1
SCHEMBL8593864 0.66 SMN1; SMN2 (0.47)
SCHEMBL6600347 0.65 MALT1 (0.35) GSK3AGSK3B
SCHEMBL8554066 0.65 TRPA1 (0.35)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096895-A Heterocyclic dihydrazole compounds and their use for controlling fungal plant diseases E. I. DU PONT DE NEMOURS AND COMPANY (US) 2000-08-01 US disclosed
EP-0825992-A1 FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1998-03-04 EP disclosed
WO-1996036633-A1 FUNGICIDAL CYCLIC AMIDES E.I. DU PONT DE NEMOURS AND COMPANY (US) 1996-11-21 WO disclosed