SCHEMBL8107948

SCHEMBL8107948

Cc1ccc(=O)n(CCN2CCN(c3cccc(C(F)(F)F)c3)CC2)n1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 5/20 0.59
SLC6A4 P31645 3/20 0.59
HTR1A P08908 6/20 0.56
HTR7 P34969 5/20 0.55
SIGMAR1 Q99720 2/20 0.54
DRD2 P14416 3/20 0.53
HTR6 P50406 1/20 0.53
ABCB11 O95342 1/20 0.53
ADRA2A P08913 1/20 0.53
ADORA3 P0DMS8 1/20 0.53
CHRM1 P11229 1/20 0.53
DRD1 P21728 1/20 0.53
TBXA2R P21731 1/20 0.53
ADRA1A P35348 1/20 0.53
OPRM1 P35372 1/20 0.53
DRD3 P35462 1/20 0.53
KCNH2 Q12809 1/20 0.53
ALDH1A1 P00352 2/20 0.52
CYP1A2 P05177 1/20 0.51
CYP3A4 P08684 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8103844 0.94 HTR2A (0.65) HTR2ASLC6A4HTR1AHTR7SIGMAR1
SCHEMBL8103442 0.94 HTR2A (0.68) HTR2ASLC6A4HTR1AHTR7SIGMAR1
SCHEMBL8103915 0.84 CTSS (0.60) HTR2ASLC6A4HTR1AHTR7SIGMAR1
SCHEMBL8102136 0.79 CTSS (0.67) HTR2ASLC6A4HTR1AHTR7SIGMAR1
SCHEMBL8103525 0.79 HTR2A (0.65) HTR2ASLC6A4HTR1AHTR7SIGMAR1
SCHEMBL7685556 0.78 KCNH2 (0.64) HTR2ASLC6A4HTR1AHTR7SIGMAR1
SCHEMBL7689489 0.78 KCNH2 (0.61) HTR2ASLC6A4HTR1AHTR7SIGMAR1
SCHEMBL2927397 0.76 ALDH1A1 (0.77) HTR1AHTR7SIGMAR1DRD2ALDH1A1
SCHEMBL11465528 0.76 SIGMAR1 (0.76) HTR2AHTR1AHTR7SIGMAR1DRD2
Ammonia Solution, Strong SCHEMBL11284383 0.75 ALDH1A1 (0.75) HTR1AHTR7SIGMAR1DRD2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1057820-A1 Arylpiperazinylalkyl-3(2H)-pyridazinones as serotonin 5HT and dopamine D2 receptor agonists FAES, Fabrica Espanola de Productos Quimicos y Farmaceuticos, S.A. (ES) 2000-12-06 EP claimed