SCHEMBL8103525

SCHEMBL8103525

O=c1ccc(-c2ccccc2)nn1CCCCN1CCN(c2cccc(C(F)(F)F)c2)CC1

nearest known ligand 0.65

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
HTR2A P28223 3/20 0.65
SLC6A4 P31645 2/20 0.65
CTSS P25774 1/20 0.65
DRD2 P14416 7/20 0.61
HTR7 P34969 5/20 0.61
HTR1A P08908 1/20 0.61
HTR6 P50406 1/20 0.61
SIGMAR1 Q99720 2/20 0.60
DRD3 P35462 6/20 0.58
ADRA1A P35348 3/20 0.58
MAPT P10636 1/20 0.56
DRD5 P21918 3/20 0.55

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8102136 0.98 CTSS (0.67) HTR2ASLC6A4CTSSDRD2HTR7
SCHEMBL8103915 0.94 CTSS (0.60) HTR2ASLC6A4CTSSDRD2HTR7
SCHEMBL8109562 0.88 DRD2 (0.58) HTR2ASLC6A4CTSSDRD2HTR7
SCHEMBL7689917 0.86 MAPT (0.73) HTR2ASLC6A4DRD2HTR7HTR1A
SCHEMBL8103442 0.85 HTR2A (0.68) HTR2ASLC6A4DRD2HTR7HTR1A
SCHEMBL7689812 0.84 MAPT (0.73) HTR2ASLC6A4CTSSDRD2HTR7
SCHEMBL8103844 0.83 HTR2A (0.65) HTR2ASLC6A4CTSSDRD2HTR7
SCHEMBL7683387 0.79 MAPT (0.72) HTR2ASLC6A4DRD2HTR7HTR1A
Hydrochloric Acid SCHEMBL8402882 0.79 DRD2 (0.57) HTR2ASLC6A4DRD2HTR7HTR1A
Hydrochloric Acid SCHEMBL8557013 0.79 DRD2 (0.62) HTR2ASLC6A4DRD2HTR7HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1057820-A1 Arylpiperazinylalkyl-3(2H)-pyridazinones as serotonin 5HT and dopamine D2 receptor agonists FAES, Fabrica Espanola de Productos Quimicos y Farmaceuticos, S.A. (ES) 2000-12-06 EP claimed