SCHEMBL8109692

SCHEMBL8109692

O=C(Cc1ccccc1)C1(C(=O)Cc2ccccc2)CNCCN1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES1 P23141 2/20 0.41
CES2 O00748 1/20 0.41
AKR1B1 P15121 1/20 0.41
CTSD P07339 1/20 0.37
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
HDAC8 Q9BY41 1/20 0.37
HDAC6 Q9UBN7 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
TSHR P16473 1/20 0.37
MAPT P10636 1/20 0.37
CRBN Q96SW2 1/20 0.36
BCHE P06276 2/20 0.36
ACHE P22303 2/20 0.36
SLC6A2 P23975 2/20 0.36
SLC6A4 P31645 2/20 0.36
SLC6A3 Q01959 2/20 0.36
FNTA P49354 1/20 0.36
FNTB P49356 1/20 0.36
SRD5A2 P31213 2/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11727966 0.72 SLC6A2 (0.39) CES1CES2AKR1B1CTSDMEN1
Phenylacetic Acid SCHEMBL27717158 0.71 AKR1B1 (0.74) CES1CES2AKR1B1MEN1KMT2A
SCHEMBL6542682 0.71 HSD11B1 (0.43) MEN1KMT2AL3MBTL1TSHRCRBN
SCHEMBL10965642 0.68 OPRM1 (0.56) CES1CES2AKR1B1MEN1KMT2A
Hydrochloric Acid SCHEMBL27628989 0.67 OPRL1 (0.40) SLC6A2SLC6A4SLC6A3
SCHEMBL7589446 0.66 KDM4E (0.31) KMT2A
SCHEMBL8392962 0.66 CES1 (0.47) CES1CES2AKR1B1MEN1KMT2A
Piperazine SCHEMBL4405486 0.66 CES2 (0.47) CES1CES2AKR1B1CTSDMEN1
Phenylacetic Acid SCHEMBL9555521 0.65 AKR1B1 (0.68) CES1CES2AKR1B1MEN1KMT2A
SCHEMBL8391946 0.65 CES1 (0.50) CES1CES2AKR1B1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691962-B1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AG (DE) 2000-09-13 EP disclosed
US-5622953-A DRUG RESISTANT TO ANTICANCER CHEMOTHERAPEUTIC DRUG BASF AKTIENGESELLSCHAFT (DE) 1997-04-22 US disclosed
EP-0691962-A1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AKTIENGESELLSCHAFT (DE) 1996-01-17 EP disclosed
WO-1994022842-A1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AKTIENGESELLSCHAFT (DE) 1994-10-13 WO disclosed