SCHEMBL8109958

SCHEMBL8109958

COCc1ccc2c(c1)CN(c1nc(Cl)nc(C)c1C)CC2

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM3 P20309 1/20 0.35
PDE4A P27815 1/20 0.35
PDE4B Q07343 1/20 0.35
PDE4C Q08493 1/20 0.35
PDE4D Q08499 1/20 0.35
ROCK2 O75116 1/20 0.35
ROCK1 Q13464 1/20 0.35
ALDH1A1 P00352 1/20 0.33
GAA P10253 1/20 0.33
RAD52 P43351 1/20 0.33
FAAH O00519 1/20 0.33
ADAMTS4 O75173 1/20 0.33
SYK P43405 1/20 0.31
KMT2A Q03164 1/20 0.31
ABCB1 P08183 1/20 0.31
ABCC1 P33527 1/20 0.31
ABCG2 Q9UNQ0 1/20 0.31
GRIN2D O15399 2/20 0.31
GRIN3B O60391 2/20 0.31
GRIN1 Q05586 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8117433 0.96 FAAH (0.35) CHRM3PDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL8117259 0.78 KCNH3 (0.38) ROCK2ROCK1RAD52KMT2A
SCHEMBL6966650 0.78 CHRM3 (0.49) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL6966656 0.76 CHRM3 (0.46) CHRM3PDE4APDE4BPDE4CPDE4D
Hydrochloric Acid SCHEMBL8111169 0.74 KCNH3 (0.38) ROCK2ROCK1RAD52KMT2A
SCHEMBL6997338 0.67 PDE4A (0.46) CHRM3PDE4APDE4BPDE4CPDE4D
SCHEMBL10071548 0.65 RXRB (0.41) ALDH1A1NPC1RAB9ASMN1; SMN2
SCHEMBL25488835 0.65 MAOB (0.51) PDE4DALDH1A1GAARAD52KMT2A
SCHEMBL10312978 0.65 NOTUM (0.55) KMT2AABCB1ABCC1NPC1RAB9A
SCHEMBL4760279 0.65 ACHE (0.55)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015444-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION, LTD. (KR) 2000-07-05 EP disclosed
WO-1998043968-A1 NOVEL PYRIMIDINE DERIVATIVES AND PROCESSES FOR THE PREPARATION THEREOF YUHAN CORPORATION (KR) 1998-10-08 WO disclosed