SCHEMBL8113309

SCHEMBL8113309

CC1=C(N)Nc2cc(C#N)ccc2O1.CC1=C(N)Nc2cc(C(F)(F)F)ccc2O1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KIF11 P52732 1/20 0.40
ACE2 Q9BYF1 1/20 0.39
DGAT1 O75907 1/20 0.36
SOAT1 P35610 1/20 0.36
KCNH2 Q12809 1/20 0.36
JUN P05412 1/20 0.36
NFKB1 P19838 1/20 0.36
NFKB2 Q00653 1/20 0.36
RELA Q04206 1/20 0.36
TDO2 P48775 1/20 0.35
PTGDR2 Q9Y5Y4 1/20 0.34
SHMT1 P34896 4/20 0.34
SCN5A Q14524 1/20 0.32
SCN9A Q15858 1/20 0.32
KIT P10721 1/20 0.32
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
ALOX15 P16050 1/20 0.32
BRCA1 P38398 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6999042 0.88 ACE2 (0.47) KIF11ACE2JUNNFKB1NFKB2
SCHEMBL7002017 0.88 ABL1 (0.35) KDM4EALDH1A1
SCHEMBL27344607 0.78 ACE2 (0.43) KIF11ACE2DGAT1SOAT1KCNH2
SCHEMBL7988325 0.76 ALDH1A1 (0.36) ACE2KCNH2JUNNFKB1NFKB2
SCHEMBL28404933 0.70 ABL1 (0.43)
SCHEMBL5671424 0.69 MMP12 (0.45) MEN1ALDH1A1ALOX15KMT2AHSD17B10
SCHEMBL27344614 0.68 KIF11 (0.41) KIF11ACE2
SCHEMBL27344285 0.67 ACE2 (0.54) KIF11ACE2JUNNFKB1NFKB2
SCHEMBL7001776 0.67 ACE2 (0.35) ACE2
Hydrochloric Acid SCHEMBL6988641 0.66 ACE2 (0.34) ACE2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1015437-A1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 2000-07-05 EP disclosed
WO-1999012915-A1 BENZOXAZINE AND BENZOTHIAZINE DERIVATIVES AND THEIR USE IN PHARMACEUTICALS SCHERING AKTIENGESELLSCHAFT (DE) 1999-03-18 WO disclosed