SCHEMBL8115491

SCHEMBL8115491

C=CCOC(=O)CCc1cccc(N)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDP1 Q9NUW8 1/20 0.45
PKM P14618 1/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
CASP1 P29466 1/20 0.45
MAOA P21397 2/20 0.44
MAOB P27338 2/20 0.44
CYP19A1 P11511 1/20 0.42
THRA P10827 1/20 0.42
THRB P10828 1/20 0.42
TSHR P16473 2/20 0.42
ALDH1A1 P00352 1/20 0.42
HSD17B10 Q99714 1/20 0.42
TRPV1 Q8NER1 1/20 0.41
APP P05067 2/20 0.41
CYP3A4 P08684 1/20 0.41
NPSR1 Q6W5P4 1/20 0.40
FFAR1 O14842 1/20 0.38
GRM2 Q14416 1/20 0.38
GRM3 Q14832 1/20 0.38
L3MBTL1 Q9Y468 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11628857 0.85 ALDH1A1 (0.48) PKMSMN1; SMN2MAOAMAOBCYP19A1
SCHEMBL5687905 0.84 OPRM1 (0.49) TDP1PKMSMN1; SMN2CASP1TRPV1
SCHEMBL250955 0.82 TDP1 (0.68) TDP1PKMSMN1; SMN2CASP1ALDH1A1
SCHEMBL1068218 0.81 CYP4F2 (0.55) TDP1SMN1; SMN2MAOAMAOBCYP19A1
SCHEMBL8104566 0.81 FAAH (0.41) TDP1PKMSMN1; SMN2CASP1MAOA
SCHEMBL6999007 0.80 CASP1 (0.46) CASP1MAOAMAOBCYP19A1TSHR
SCHEMBL5450328 0.79 TDP1 (0.56) TDP1CASP1MAOAMAOBCYP19A1
Hydrochloric Acid SCHEMBL3021844 0.79 CYP4F2 (0.54) TDP1SMN1; SMN2MAOAMAOBCYP19A1
SCHEMBL7781858 0.79 APP (0.51) TDP1PKMSMN1; SMN2CASP1CYP19A1
SCHEMBL16016129 0.79 MAOB (0.52) TDP1SMN1; SMN2MAOAMAOBCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0590885-B1 Antibiotic carbapenem compounds ZENECA LTD (GB) 2000-03-15 EP disclosed
US-5527791-A Carbapenem antibiotic compounds ZENECA LIMITED (GB) 1996-06-18 US disclosed
EP-0590885-A1 Antibiotic carbapenem compounds ZENECA LIMITED (GB) 1994-04-06 EP disclosed
EP-0077662-B1 PREPARATION OF NITROARYLACETIC ACID ESTERS AND DERIVATIVES THEREOF ETHYL CORPORATION (US) 1985-10-02 EP disclosed