SCHEMBL8104566

SCHEMBL8104566

C=CCOC(=O)COCc1cccc(N)c1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FAAH O00519 2/20 0.41
ALDH1A1 P00352 3/20 0.40
HSD17B10 Q99714 3/20 0.40
TSHR P16473 2/20 0.40
TDP1 Q9NUW8 1/20 0.40
CYP3A4 P08684 1/20 0.39
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
PKM P14618 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
KDM4E B2RXH2 3/20 0.36
HPGD P15428 2/20 0.36
MAOB P27338 3/20 0.35
MAOA P21397 2/20 0.35
HCAR2 Q8TDS4 1/20 0.35
CYP19A1 P11511 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
CASP1 P29466 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11628857 0.83 ALDH1A1 (0.48) ALDH1A1HSD17B10TSHRCYP3A4THRA
SCHEMBL8228724 0.83 FAAH (0.54) FAAHALDH1A1HSD17B10TSHRTDP1
SCHEMBL823910 0.81 MAOB (0.44) ALDH1A1TSHRTDP1CYP3A4THRA
SCHEMBL8115491 0.81 TDP1 (0.45) ALDH1A1HSD17B10TSHRTDP1CYP3A4
SCHEMBL8112886 0.80 RAB9A (0.48) ALDH1A1TSHRKDM4EMAOBMAOA
SCHEMBL8116474 0.78 ALDH1A1 (0.50) ALDH1A1HSD17B10TSHRCYP3A4NPSR1
SCHEMBL15152717 0.76 THRA (0.51) ALDH1A1TDP1THRATHRBMAOB
SCHEMBL6746646 0.75 THRA (0.44) ALDH1A1TDP1THRATHRBMAOB
SCHEMBL6999007 0.72 CASP1 (0.46) FAAHALDH1A1HSD17B10TSHRMAOB
SCHEMBL366865 0.72 MAOB (0.56) ALDH1A1TSHRTDP1CYP3A4THRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0590885-B1 Antibiotic carbapenem compounds ZENECA LTD (GB) 2000-03-15 EP disclosed
US-5527791-A Carbapenem antibiotic compounds ZENECA LIMITED (GB) 1996-06-18 US disclosed
EP-0590885-A1 Antibiotic carbapenem compounds ZENECA LIMITED (GB) 1994-04-06 EP disclosed