SCHEMBL8117201

SCHEMBL8117201

O=C1C=NC(c2cccc(Cl)c2)=N1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 1/20 0.42
NOTUM Q6P988 3/20 0.41
MAOB P27338 1/20 0.39
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
NFKB1 P19838 1/20 0.39
RAB9A P51151 1/20 0.39
NFKB2 Q00653 1/20 0.39
RELA Q04206 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
ALOX5 P09917 1/20 0.38
IDO1 P14902 4/20 0.38
PGR P06401 1/20 0.37
TAAR1 Q96RJ0 1/20 0.37
KDM1A O60341 1/20 0.37
MAOA P21397 1/20 0.37
CHRNB4 P30926 1/20 0.37
CHRNA3 P32297 1/20 0.37
KDM4E B2RXH2 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10628315 0.79 MAOA (0.44) BRD4TSHRMAOAKDM4EALDH1A1
SCHEMBL643335 0.77 MAPT (0.37) NOTUMNPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL27943422 0.70 IKBKE (0.42) NOTUMNPC1TP53TSHRNFKB1
SCHEMBL8620821 0.68
SCHEMBL31222672 0.68 ALOX5 (0.65) NOTUMMAOBNPC1TP53TSHR
SCHEMBL817554 0.68 ALOX5 (0.65) NOTUMMAOBNPC1TP53TSHR
Hydrochloric Acid SCHEMBL31070804 0.66 ALOX5 (0.62) NOTUMMAOBNPC1TP53TSHR
SCHEMBL29629014 0.66 ALOX5 (0.62) NOTUMMAOBNPC1TP53TSHR
Hydrochloric Acid SCHEMBL28332867 0.66 ALOX5 (0.62) NOTUMMAOBNPC1TP53TSHR
SCHEMBL8043972 0.66 ALDH1A1 (0.45) NOTUMNPC1TP53TSHRNFKB1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042325-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE Takeda Chemical Industries, Ltd. (JP) 2000-10-11 EP disclosed
WO-1999033831-A1 NITROGEN-CONTAINING HETEROCYCLIC COMPOUNDS, THEIR PRODUCTION AND USE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1999-07-08 WO disclosed