SCHEMBL8123268

SCHEMBL8123268

O=C1Nc2ccccc2[C]c2ccccc21

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LRRK2 Q5S007 3/20 0.55
ACVR1 Q04771 2/20 0.55
PDGFRA P16234 1/20 0.55
FER P16591 1/20 0.55
LTK P29376 1/20 0.55
CDK8 P49336 1/20 0.55
DYRK1B Q9Y463 1/20 0.55
MAOA P21397 1/20 0.50
MAOB P27338 1/20 0.50
GSK3B P49841 3/20 0.48
L3MBTL1 Q9Y468 1/20 0.47
SMN1; SMN2 Q16637 3/20 0.44
CYP1A2 P05177 1/20 0.44
CSNK1G1 Q9HCP0 1/20 0.42
CHEK1 O14757 1/20 0.42
CASP3 P42574 1/20 0.42
CASP2 P42575 1/20 0.42
CASP7 P55210 1/20 0.42
CASP6 P55212 1/20 0.42
CASP8 Q14790 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL12319785 0.84 LRRK2 (0.55) LRRK2ACVR1PDGFRAFERLTK
SCHEMBL302509 0.79 MAOA (0.37) LRRK2ACVR1PDGFRAFERLTK
SCHEMBL577541 0.78 GAA (0.43) LRRK2ACVR1PDGFRAFERLTK
SCHEMBL577542 0.78 GAA (0.43) LRRK2ACVR1PDGFRAFERLTK
SCHEMBL3942970 0.76 LRRK2 (0.45) LRRK2ACVR1PDGFRAFERLTK
SCHEMBL2420711 0.75 LRRK2 (0.90) LRRK2ACVR1PDGFRAFERLTK
SCHEMBL366728 0.75
SCHEMBL1368292 0.72 LRRK2 (1.00) LRRK2ACVR1PDGFRAFERLTK
SCHEMBL27980501 0.72 LRRK2 (0.82) LRRK2ACVR1PDGFRAFERLTK
SCHEMBL27425410 0.72 LRRK2 (0.74) LRRK2ACVR1PDGFRAFERLTK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6114390-A AN ARGININAMIDE OR ORNITHINAMIDE COMPOUND AS TREATING MEMORY LOSS, MIGRAINE, SLEEP DISORDERS, PAIN, CARDIOVASCULAR DISEASES, SUBARACHNOIDAL BLEEDING, VASCULAR-HYPERTROPHIC CHANGES, CEREBRAL AND CORONARY VASOSPASMS KARL THOMAE GMBH (DE) 2000-09-05 US disclosed
EP-0680469-B1 AMINOACID DERIVATES, MEDICAMENTS CONTAINING THESE COMPOUNDS AND PROCESS FOR PREPARING THE SAME BOEHRINGER INGELHEIM PHARMA (DE) 2000-04-26 EP disclosed
US-5616620-A HYPOTENSIVE AGENTS KARL THOMAE GMBH (DE) 1997-04-01 US disclosed