SCHEMBL8133019

SCHEMBL8133019

O=C(O)C(Br)c1ccccc1Br

nearest known ligand 0.45

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CES2 O00748 2/20 0.45
CES1 P23141 2/20 0.45
HTT P42858 2/20 0.42
CYP1A2 P05177 1/20 0.41
IDO1 P14902 1/20 0.40
TDO2 P48775 1/20 0.40
SRC P12931 2/20 0.38
CYP2D6 P10635 1/20 0.38
LMNA P02545 3/20 0.37
MAPK1 P28482 1/20 0.37
OPRL1 P41146 1/20 0.37
CYP2C9 P11712 1/20 0.36
CYP2C19 P33261 1/20 0.36
MEN1 O00255 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
KMT2A Q03164 1/20 0.36
HSD11B1 P28845 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8133022 1.00 CES2 (0.45) CES2CES1HTTCYP1A2IDO1
SCHEMBL20930584 0.84 CYP2D6 (0.50) CES2CES1HTTCYP1A2IDO1
SCHEMBL6046964 0.80 CES2 (0.39) CES2CES1HTTCYP1A2IDO1
SCHEMBL11577707 0.80 HTT (0.43) CES2CES1HTTCYP1A2IDO1
SCHEMBL196781 0.78 LMNA (0.52) CES2CES1HTTCYP1A2IDO1
SCHEMBL30670484 0.78 LMNA (0.52) CES2CES1HTTCYP1A2IDO1
SCHEMBL8127769 0.78 LMNA (0.52) CES2CES1HTTCYP1A2IDO1
SCHEMBL196782 0.78 LMNA (0.52) CES2CES1HTTCYP1A2IDO1
SCHEMBL27765065 0.78 GABRA1 (0.46) CES2CES1CYP1A2SRCCYP2D6
SCHEMBL17673198 0.78 HTT (0.46) HTTCYP1A2IDO1TDO2CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6124343-A Substituted phenyl compounds with a substituent having a thienyl ring RHONE-POULENC RORER LIMITED (GB) 2000-09-26 US disclosed
EP-0805802-B1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE POULENC RORER LTD (GB) 2000-08-16 EP disclosed
US-6048893-A Substituted phenyl compounds with a substituent having A 1,3-benzodioxole ring RHONE-POULENC RORER LIMITED (GB) 2000-04-11 US disclosed
EP-0805802-A1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE-POULENC RORER LIMITED (GB) 1997-11-12 EP disclosed
WO-1996022978-A1 SUBSTITUTED PHENYL COMPOUNDS AS ENDOTHELIN ANTAGONISTS RHONE POULENC RORER LIMITED (GB) 1996-08-01 WO disclosed