SCHEMBL8149484

SCHEMBL8149484

CN1CCC(c2n[nH]c3ccc(NC(=O)Nc4ccccc4)cc23)CC1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TP53 P04637 1/20 0.48
MAPT P10636 1/20 0.48
HTR1D P28221 12/20 0.48
HTR1B P28222 12/20 0.48
HTR1F P30939 3/20 0.48
HTR1A P08908 2/20 0.48
ITK Q08881 1/20 0.48
AURKA O14965 1/20 0.47
DYRK1A Q13627 1/20 0.47
TTK P33981 1/20 0.47
ROCK2 O75116 1/20 0.45
ROCK1 Q13464 1/20 0.45
CA12 O43570 1/20 0.44
CA9 Q16790 1/20 0.44
BRD4 O60885 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8154553 0.89 NPC1 (0.47) TP53MAPTHTR1AITKAURKA
SCHEMBL5906202 0.85 HTR1D (0.44) HTR1DHTR1BHTR1FHTR1ADYRK1A
SCHEMBL8148939 0.82 ULK1 (0.44) ITKAURKATTKROCK2ROCK1
SCHEMBL8148201 0.81 ULK1 (0.44) ITKAURKATTKROCK2ROCK1
SCHEMBL5315176 0.81 HTR1D (0.69) HTR1DHTR1BHTR1FHTR1A
SCHEMBL3147519 0.80 HTR6 (0.60) ITKAURKABRD4
SCHEMBL7481815 0.80 HTR1D (0.76) MAPTHTR1DHTR1BHTR1FHTR1A
SCHEMBL8146828 0.79 DRD2 (0.43) MAPT
Hydrochloric Acid SCHEMBL7489449 0.79 HTR1D (0.74) MAPTHTR1DHTR1BHTR1FHTR1A
SCHEMBL5309846 0.79 HTR1D (0.52) MAPTHTR1DHTR1BHTR1FHTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000006173-A1 5-HT1F AGONISTS ELI LILLY AND COMPANY (US) 2000-02-10 WO disclosed