SCHEMBL8150307

SCHEMBL8150307

COc1ccc([CH]CC(C)C)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
CYP2A6 P11509 1/20 0.54
KDM4E B2RXH2 3/20 0.47
LMNA P02545 2/20 0.47
CYP3A4 P08684 2/20 0.47
TP53 P04637 1/20 0.47
TSHR P16473 1/20 0.47
CA12 O43570 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
CA7 P43166 1/20 0.46
CA9 Q16790 1/20 0.46
CA14 Q9ULX7 1/20 0.46
TRPA1 O75762 1/20 0.45
RELA Q04206 1/20 0.45
TDP1 Q9NUW8 1/20 0.44
ESR1 P03372 2/20 0.44
CYP1A2 P05177 2/20 0.44
ABL1 P00519 1/20 0.44
TTR P02766 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6320160 0.84 TYR (0.39) ALDH1A1CYP2A6
SCHEMBL8325507 0.78 TRPA1 (0.50) ALDH1A1CYP2A6TRPA1
SCHEMBL1004990 0.78 ALDH1A1 (0.62) ALDH1A1CYP2A6KDM4ELMNACYP3A4
SCHEMBL1253022 0.74 ALDH1A1 (0.58) ALDH1A1CYP2A6KDM4ELMNACYP3A4
SCHEMBL3350071 0.74 ALDH1A1 (0.58) ALDH1A1CYP2A6KDM4ELMNACYP3A4
SCHEMBL3184498 0.74 ALDH1A1 (0.58) ALDH1A1CYP2A6KDM4ELMNACYP3A4
SCHEMBL436098 0.74 HSD17B10 (0.46) ALDH1A1CYP2A6LMNATRPA1CYP1A2
SCHEMBL8321285 0.73 TRPA1 (0.49) ALDH1A1CYP2A6KDM4ETRPA1CYP1A2
SCHEMBL3422525 0.73 ALDH1A1 (0.47) ALDH1A1CYP2A6KDM4ELMNACYP3A4
SCHEMBL543436 0.73 HTR2A (0.47) ALDH1A1CYP2A6LMNACYP3A4TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6147061-A ANTIARTHRITIC AGENTS; ANTICANCER AGENTS; ORAL DISEASES PFIZER INC. (US) 2000-11-14 US disclosed
EP-0821669-A1 HYDROXAMIC AND CARBOXYLIC ACIDS AS METALLOPROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-02-04 EP disclosed
US-5691381-A ANTAGONIST OF TUMOR NECROSIS FACTOR, ANTIINFLAMMATORY AGENT, ANTIARTHRITIC AGENT THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-25 US disclosed