SCHEMBL8155829

SCHEMBL8155829

O=C1NCCc2cc(-c3ccccc3F)ccc21

nearest known ligand 0.68

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP11 Q9NR21 10/20 0.68
PARP10 Q53GL7 10/20 0.68
GRM5 P41594 5/20 0.59
PARP1 P09874 3/20 0.58
PDPK1 O15530 1/20 0.58
PTPRC P08575 1/20 0.50
PTPN1 P18031 1/20 0.50
HRH3 Q9Y5N1 1/20 0.49
PLK4 O00444 1/20 0.48
MAPK13 O15264 1/20 0.48
DAPK3 O43293 1/20 0.48
DYRK3 O43781 1/20 0.48
RPS6KA4 O75676 1/20 0.48
PRKD3 O94806 1/20 0.48
MAP4K4 O95819 1/20 0.48
CHEK2 O96017 1/20 0.48
EGFR P00533 1/20 0.48
CDK1 P06493 1/20 0.48
MET P08581 1/20 0.48
PIM1 P11309 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18113016 0.86 MAPK1 (0.57) PARP11PARP10GRM5PARP1PDPK1
SCHEMBL8151102 0.85 PARP10 (0.70) PARP11PARP10GRM5PARP1PDPK1
SCHEMBL8167365 0.82 PARP11 (0.68) PARP11PARP10GRM5PARP1PDPK1
SCHEMBL8154134 0.82 PARP11 (0.68) PARP11PARP10GRM5PARP1PDPK1
SCHEMBL8155722 0.81 PARP11 (1.00) PARP11PARP10GRM5PARP1PDPK1
SCHEMBL8167145 0.80 PARP10 (0.76) PARP11PARP10GRM5PARP1PDPK1
SCHEMBL20294385 0.79 PARP11 (0.72) PARP11PARP10GRM5PARP1PDPK1
SCHEMBL8151110 0.79 PARP10 (0.78) PARP11PARP10GRM5PARP1PDPK1
SCHEMBL8633556 0.78 HSD17B1 (0.60) GRM5PARP1PTPRCPTPN1HRH3
SCHEMBL8163095 0.78 GSK3B (0.74) PARP11PARP10GRM5PARP1PDPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008151184-A1 BENZAMIDE MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2008-12-11 WO disclosed