SCHEMBL8633556

SCHEMBL8633556

O=C1CCc2cc(-c3ccccc3F)ccc21

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B1 P14061 4/20 0.60
PTPRC P08575 1/20 0.56
PTPN1 P18031 1/20 0.56
HRH3 Q9Y5N1 1/20 0.53
PARP1 P09874 1/20 0.53
PARP2 Q9UGN5 1/20 0.53
CYP11B1 P15538 2/20 0.51
CYP11B2 P19099 2/20 0.51
CYP1A2 P05177 1/20 0.51
GRM5 P41594 1/20 0.47
CASP1 P29466 1/20 0.47
CASP7 P55210 1/20 0.47
HSD17B10 Q99714 1/20 0.47
DHODH Q02127 1/20 0.44
ACMSD Q8TDX5 1/20 0.43
ADORA1 P30542 1/20 0.43
PGR P06401 1/20 0.43
TNKS O95271 1/20 0.42
TNKS2 Q9H2K2 1/20 0.42
CYP2A6 P11509 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8072264 0.90 HRH3 (0.54) HSD17B1PTPRCPTPN1HRH3PARP1
SCHEMBL8635876 0.90 HSD17B1 (0.56) HSD17B1PTPRCPTPN1HRH3PARP1
SCHEMBL8631353 0.87 PTPRC (0.56) HSD17B1PTPRCPTPN1HRH3PARP1
SCHEMBL5937022 0.80 HSD17B1 (0.63) HSD17B1CYP11B1CYP11B2CYP1A2GRM5
SCHEMBL8635273 0.80 PTPRC (0.46) HSD17B1PTPRCPTPN1HRH3PARP1
SCHEMBL8635928 0.80 PARP1 (0.48) HSD17B1PTPRCPTPN1HRH3PARP1
SCHEMBL28655414 0.80 HSD17B1 (0.78) HSD17B1HRH3CYP11B1CYP11B2CYP1A2
SCHEMBL28841436 0.80 HSD17B1 (0.50) HSD17B1CYP11B1CYP11B2CYP1A2GRM5
SCHEMBL1745161 0.79 HSD17B1 (0.71) HSD17B1HRH3CYP11B1CYP11B2CYP1A2
SCHEMBL8155829 0.78 PARP11 (0.68) PTPRCPTPN1HRH3PARP1PARP2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0601191-B1 NOVEL TETRACYCLIC COMPOUND KYOWA HAKKO KOGYO KK (JP) 1998-07-22 EP disclosed
US-5371225-A Immunosuppressants KYOWA HAKKO KOGYO CO., LTD. (JP) 1994-12-06 US disclosed
EP-0601191-A1 NOVEL TETRACYCLIC COMPOUND KYOWA HAKKO KOGYO KABUSHIKI KAISHA (JP) 1994-06-15 EP disclosed