SCHEMBL8163095

SCHEMBL8163095

Cc1cc(-c2ccc3c(c2)CCNC3=O)ccc1F

nearest known ligand 0.74

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 2/20 0.74
DAPK3 O43293 1/20 0.74
NTRK1 P04629 1/20 0.74
PIM1 P11309 1/20 0.74
FLT3 P36888 1/20 0.74
ROCK1 Q13464 1/20 0.74
CLK4 Q9HAZ1 1/20 0.74
GRM5 P41594 6/20 0.70
PARP10 Q53GL7 11/20 0.64
PARP11 Q9NR21 10/20 0.64
PARP1 P09874 3/20 0.48
PDPK1 O15530 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8154044 0.83 DAPK3 (0.55) GSK3BDAPK3NTRK1PIM1FLT3
SCHEMBL504652 0.82 GRM5 (1.00) GSK3BDAPK3NTRK1PIM1FLT3
SCHEMBL8167145 0.82 PARP10 (0.76) GSK3BDAPK3NTRK1PIM1FLT3
SCHEMBL16561672 0.82 PARP10 (0.76) GSK3BDAPK3NTRK1PIM1FLT3
SCHEMBL8151110 0.81 PARP10 (0.78) GSK3BDAPK3NTRK1PIM1FLT3
SCHEMBL8155836 0.79 PARP10 (0.76) GSK3BNTRK1FLT3GRM5PARP10
SCHEMBL12559528 0.79 GRM5 (0.59) GSK3BDAPK3NTRK1PIM1FLT3
SCHEMBL8156296 0.78 PARP10 (1.00) GSK3BCLK4GRM5PARP10PARP11
SCHEMBL8151102 0.78 PARP10 (0.70) GSK3BDAPK3NTRK1PIM1FLT3
SCHEMBL8155829 0.78 PARP11 (0.68) DAPK3PIM1CLK4GRM5PARP10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008151184-A1 BENZAMIDE MGLUR5 POSITIVE ALLOSTERIC MODULATORS AND METHODS OF MAKING AND USING SAME VANDERBILT UNIVERSITY (US) 2008-12-11 WO disclosed