SCHEMBL8159852

SCHEMBL8159852

CCOC(=O)c1[nH]c2ccccc2c1-n1c(-c2cn(C)c3ccccc23)c[nH]c1=O

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 7/20 0.46
MAPT P10636 2/20 0.46
NPSR1 Q6W5P4 1/20 0.46
HPGD P15428 3/20 0.45
TSHR P16473 1/20 0.45
HSD17B10 Q99714 1/20 0.45
GAA P10253 2/20 0.44
NPC1 O15118 1/20 0.44
SMN1; SMN2 Q16637 1/20 0.44
KDM4E B2RXH2 10/20 0.44
HTR6 P50406 2/20 0.42
TUBB4A P04350 2/20 0.41
TUBB P07437 2/20 0.41
TUBA3C P0DPH7 2/20 0.41
TUBA1B P68363 2/20 0.41
TUBA4A P68366 2/20 0.41
TUBB4B P68371 2/20 0.41
TUBB3 Q13509 2/20 0.41
TUBB2A Q13885 2/20 0.41
TUBB8 Q3ZCM7 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7008865 0.77 PIM1 (0.40) CCNT1PIM1CDK9
SCHEMBL7507655 0.75 GAA (0.47) ALDH1A1MAPTNPSR1HPGDTSHR
SCHEMBL7005539 0.72 CDK4 (0.55) ALDH1A1MAPTHPGDTSHRHSD17B10
SCHEMBL7005313 0.72 PKM (0.40) ALDH1A1MAPTNPSR1HPGDGAA
SCHEMBL7005879 0.70 PIM1 (0.48) MAPTTSHRHSD17B10SMN1; SMN2MEN1
Acetic Acid SCHEMBL7011660 0.68 CAMK2D (0.46) MAPTTSHRHSD17B10SMN1; SMN2MEN1
SCHEMBL7010209 0.68 PIM1 (0.37) MAPTTSHRHSD17B10SMN1; SMN2MEN1
SCHEMBL7008320 0.67 RPS6KB1 (0.41) ALDH1A1MAPTTSHRGAANPC1
SCHEMBL6379635 0.67 NR4A2 (0.69) ALDH1A1MAPTNPSR1TSHRKDM4E
SCHEMBL8159849 0.67 AHR (0.41) ALDH1A1MAPTNPSR1HPGDTSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1042317-A1 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS AstraZeneca AB (SE) 2000-10-11 EP disclosed
WO-1999032483-A1 NEW PHARMACEUTICALLY ACTIVE COMPOUNDS ASTRAZENECA AB (SE) 1999-07-01 WO disclosed