SCHEMBL8161985

SCHEMBL8161985

Cc1cccc(-c2c(C(=O)c3ccc(O)cc3)ccc3cc(O)ccc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 4/20 0.47
CNR1 P21554 2/20 0.47
HSD17B1 P14061 4/20 0.43
HSD17B2 P37059 4/20 0.43
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2B6 P20813 1/20 0.41
CYP2C19 P33261 1/20 0.41
KMT2A Q03164 4/20 0.41
ESR1 P03372 2/20 0.41
CA12 O43570 1/20 0.41
CA9 Q16790 1/20 0.41
NPC1 O15118 3/20 0.40
RAB9A P51151 2/20 0.40
MEN1 O00255 2/20 0.40
CLK1 P49759 1/20 0.40
DYRK1A Q13627 1/20 0.40
DYRK1B Q9Y463 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8165414 0.86 ESR1 (0.52) CNR2CNR1HSD17B1HSD17B2KMT2A
SCHEMBL11620607 0.85 MEN1 (0.53) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL11621961 0.81 MEN1 (0.55) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL9301900 0.81 HSD17B1 (0.43) CNR2CNR1HSD17B1HSD17B2CYP1A2
SCHEMBL8160039 0.80 CLK1 (0.50) HSD17B1HSD17B2CYP1A2CYP3A4CYP2D6
SCHEMBL8153524 0.77 KMT2A (0.46) CYP3A4KMT2AESR1NPC1RAB9A
SCHEMBL8339441 0.76 CNR2 (0.59) CNR2CNR1HSD17B1HSD17B2KMT2A
SCHEMBL8160201 0.76 MEN1 (0.44) KMT2AESR1NPC1RAB9AMEN1
SCHEMBL8338455 0.74 ESR1 (0.66) CNR2CNR1HSD17B1HSD17B2ESR1
SCHEMBL8160628 0.72 MMP2 (0.47) CYP3A4KMT2AESR1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6107346-A ADMINISTERING AND AROMATIC KETONE COMPOUND ELI LILLY AND COMPANY (US) 2000-08-22 US disclosed
EP-0897903-A2 Ketone-derivatives of indene, dihydronaphthalene or naphthalene compounds for the treatment of hyperlipidemia ELI LILLY AND COMPANY (US) 1999-02-24 EP disclosed
WO-1999007360-A1 COMPOUNDS AND USES THEREOF ELI LILLY AND COMPANY (US) 1999-02-18 WO disclosed