SCHEMBL8167606

SCHEMBL8167606

CCN(Cc1cc(Br)ccc1OCc1ccc(Cl)cc1)c1ccc(C(=O)O)cn1

nearest known ligand 0.58

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 11/20 0.58
PTGER1 P34995 3/20 0.52
MRGPRX4 Q96LA9 2/20 0.48
STAT3 P40763 1/20 0.45
NPSR1 Q6W5P4 1/20 0.45
RXRA P19793 1/20 0.44
XDH P47989 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8703967 0.94 CCR5 (0.48) CCR5PTGER1RXRAXDH
SCHEMBL8701112 0.91 CCR5 (0.46) CCR5PTGER1RXRAXDH
SCHEMBL1907786 0.91 RXRA (0.53) CCR5PTGER1RXRA
SCHEMBL8161455 0.90 PTGER1 (0.54) CCR5PTGER1MRGPRX4RXRA
SCHEMBL8162210 0.90 ALDH1A1 (0.45) CCR5PTGER1NPSR1RXRAXDH
SCHEMBL8163058 0.87 RXRA (0.53) PTGER1MRGPRX4RXRA
SCHEMBL8167611 0.87 CCR5 (0.56) CCR5PTGER1STAT3NPSR1
SCHEMBL7672615 0.84 HCAR3 (0.51) RXRA
SCHEMBL7963005 0.84 HCAR3 (0.44) CCR5RXRA
SCHEMBL7963047 0.84 HCAR3 (0.44) CCR5RXRA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773930-B1 AROMATIC AMINO ETHERS AS PAIN RELIEVING AGENTS ZENECA LTD (GB) 2000-10-11 EP claimed
US-5843942-A Aromatic amino ethers as pain relieving agents ZENECA LIMITED (GB) 1998-12-01 US disclosed
EP-0773930-A1 AROMATIC AMINO ETHERS AS PAIN RELIEVING AGENTS ZENECA LIMITED (GB) 1997-05-21 EP disclosed
WO-1996003380-A1 AROMATIC AMINO ETHERS AS PAIN RELIEVING AGENTS ZENECA LIMITED (GB) 1996-02-08 WO disclosed