SCHEMBL8701112

SCHEMBL8701112

CCN(Cc1cc(Br)ccc1OCc1ccc(C)cc1)c1ccc(C(=O)O)cn1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 4/20 0.46
RXRA P19793 1/20 0.45
XDH P47989 2/20 0.45
PTGER1 P34995 10/20 0.44
HCAR3 P49019 1/20 0.44
CYP1A2 P05177 2/20 0.43
HTR7 P34969 1/20 0.43
HTR6 P50406 1/20 0.43
NPC1 O15118 1/20 0.41
ALDH1A1 P00352 1/20 0.41
LMNA P02545 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
MAPT P10636 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
RECQL P46063 1/20 0.41
RAB9A P51151 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8703967 0.95 CCR5 (0.48) CCR5RXRAXDHPTGER1HCAR3
SCHEMBL1907786 0.92 RXRA (0.53) CCR5RXRAPTGER1HCAR3CYP1A2
SCHEMBL8167606 0.91 CCR5 (0.58) CCR5RXRAXDHPTGER1
SCHEMBL8162210 0.90 ALDH1A1 (0.45) CCR5RXRAXDHPTGER1HCAR3
SCHEMBL8161455 0.85 PTGER1 (0.54) CCR5RXRAPTGER1
SCHEMBL7672615 0.85 HCAR3 (0.51) RXRAHCAR3NPC1LMNAMAPT
SCHEMBL8167295 0.85 PTGER1 (0.46) CCR5RXRAPTGER1CYP1A2ALDH1A1
SCHEMBL6256530 0.84 RXRA (0.51) CCR5RXRAPTGER1HCAR3CYP1A2
SCHEMBL7662467 0.84 CCR5 (0.45) CCR5RXRAPTGER1CYP1A2ALDH1A1
SCHEMBL8167287 0.83 HCAR3 (0.41) CCR5RXRAPTGER1HCAR3CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0773930-A1 AROMATIC AMINO ETHERS AS PAIN RELIEVING AGENTS ZENECA LIMITED (GB) 1997-05-21 EP claimed
US-5843942-A Aromatic amino ethers as pain relieving agents ZENECA LIMITED (GB) 1998-12-01 US disclosed
WO-1996003380-A1 AROMATIC AMINO ETHERS AS PAIN RELIEVING AGENTS ZENECA LIMITED (GB) 1996-02-08 WO disclosed