SCHEMBL8168565

SCHEMBL8168565

Nc1cccnc1N1CCN(C(=O)Cc2ccc(OC3CCOC3)cc2)CC1

nearest known ligand 0.45

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HPGD P15428 2/20 0.45
HSD17B10 Q99714 2/20 0.45
NPSR1 Q6W5P4 1/20 0.45
L3MBTL1 Q9Y468 1/20 0.45
KDM4E B2RXH2 4/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
GRM4 Q14833 2/20 0.39
IDH1 O75874 1/20 0.39
RBP4 P02753 1/20 0.39
FFAR4 Q5NUL3 1/20 0.38
ALDH1A1 P00352 2/20 0.37
CPT2 P23786 2/20 0.37
CPT1A P50416 2/20 0.37
AKT1 P31749 1/20 0.37
GFER P55789 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3339826 0.87 KDM4E (0.55) HPGDHSD17B10NPSR1L3MBTL1KDM4E
SCHEMBL8167199 0.78 ME2 (0.54) HPGDHSD17B10NPSR1L3MBTL1KDM4E
SCHEMBL8168851 0.78 SLC6A7 (0.53) HPGDHSD17B10NPSR1L3MBTL1KDM4E
SCHEMBL8168338 0.76 SLC6A7 (0.55) HPGDHSD17B10NPSR1L3MBTL1KDM4E
SCHEMBL8163504 0.72 PANK3 (0.48) HPGDHSD17B10NPSR1L3MBTL1KDM4E
SCHEMBL8172191 0.70 KDM4E (0.45) HPGDHSD17B10NPSR1L3MBTL1KDM4E
SCHEMBL1812295 0.69 ACACB (0.45)
SCHEMBL1812294 0.69 ACACB (0.45)
SCHEMBL3333923 0.68 KDM4E (0.62) KDM4ESMN1; SMN2RBP4ALDH1A1
SCHEMBL3334455 0.67 TRPA1 (0.55) HPGDHSD17B10NPSR1L3MBTL1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008112440-A1 PIPERAZINE AND PIPERIDINE MGLUR5 POTENTIATORS ASTRAZENECA AB (SE) 2008-09-18 WO disclosed