SCHEMBL8173299

SCHEMBL8173299

CCCCN1CCCCC(NC(=O)c2nn(CCC)c3ccccc23)CCC1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3A P46098 6/20 0.54
HTR4 Q13639 5/20 0.53
CNR1 P21554 4/20 0.49
CNR2 P34972 4/20 0.49
MEN1 O00255 1/20 0.49
ALDH1A1 P00352 1/20 0.49
CYP1A2 P05177 1/20 0.49
CYP3A4 P08684 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
HTT P42858 1/20 0.49
KMT2A Q03164 1/20 0.49
HTR3E A5X5Y0 1/20 0.46
SLC22A2 O15244 1/20 0.46
HTR3B O95264 1/20 0.46
CHRNB2 P17787 1/20 0.46
CHRNA3 P32297 1/20 0.46
CHRNA4 P43681 1/20 0.46
KCNH2 Q12809 1/20 0.46
HTR3D Q70Z44 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6947363 0.98 HTR3A (0.56) HTR3AHTR4CNR1CNR2MEN1
SCHEMBL8172300 0.96 HTR4 (0.57) HTR3AHTR4CNR1CNR2MEN1
SCHEMBL6948706 0.92 HTR4 (0.58) HTR3AHTR4CNR1CNR2F10
SCHEMBL8173282 0.90 HTR3A (0.57) HTR3AHTR4CNR1CNR2MEN1
SCHEMBL8173531 0.89 HTR3A (0.53) HTR3AHTR4MEN1ALDH1A1CYP1A2
SCHEMBL6956463 0.88 HTR3A (0.59) HTR3AHTR4CNR1CNR2MEN1
SCHEMBL6950822 0.86 HTR3A (0.55) HTR3AHTR4MEN1ALDH1A1CYP1A2
SCHEMBL8162100 0.86 HTR3A (0.57) HTR3AHTR4CNR1CNR2MEN1
SCHEMBL8169133 0.85 HTR4 (0.54) HTR3AHTR4MEN1KMT2AF10
SCHEMBL6953090 0.84 HTR3A (0.59) HTR3AHTR4CNR1CNR2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6096746-A Indazole compound containing a monocyclic amine structure NISSHIN FLOUR MILLING CO., LTD. (JP) 2000-08-01 US disclosed
US-5945434-A TREATMENT OF GASTROINTESTINAL DISORDERS NISSHIN FLOUR MILLING CO., LTD. (JP) 1999-08-31 US disclosed
EP-0829474-A1 INDAZOLE DERIVATIVES HAVING MONOCYCLIC AMINO GROUP NISSHIN FLOUR MILLING CO., LTD. (JP) 1998-03-18 EP disclosed