SCHEMBL8183264

SCHEMBL8183264

COC(=O)C[C@H](NC(=O)OCc1ccccc1)C(=O)N(Cc1cc(C(=O)O)ccc1F)CC(F)(F)F

nearest known ligand 0.47

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
CTSL P07711 2/20 0.40
CTSB P07858 2/20 0.40
CTSS P25774 2/20 0.40
CTSK P43235 2/20 0.40
KYNU Q16719 1/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
ALDH1A1 P00352 1/20 0.39
KMT2A Q03164 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8183267 1.00 CTSL (0.40) CTSLCTSBCTSSCTSKKYNU
SCHEMBL6954036 0.87 MEN1 (0.48) CTSLCTSBCTSSCTSKKYNU
SCHEMBL6954031 0.87 MEN1 (0.48) CTSLCTSBCTSSCTSKKYNU
SCHEMBL8327721 0.83 CYP3A4 (0.43) CTSLCTSBALDH1A1
SCHEMBL12604584 0.81 SYK (0.42) CTSLCTSBCTSSCTSK
SCHEMBL4027455 0.80 LPAR1 (0.43) CTSLCTSBCTSSCTSKKYNU
SCHEMBL4027452 0.80 LPAR1 (0.43) CTSLCTSBCTSSCTSKKYNU
SCHEMBL6954041 0.79 CASP1 (0.44)
SCHEMBL6954029 0.79 CASP1 (0.44)
SCHEMBL8178607 0.79 LPAR1 (0.37) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6159964-A Vitronectin receptor antagonists SMITHKLINE BEECHAM CORPORATION (US) 2000-12-12 US disclosed
EP-0906103-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1999-04-07 EP disclosed
EP-0906103-A4 1999-04-07 EP disclosed
WO-1997024124-A1 VITRONECTIN RECEPTOR ANTAGONISTS SMITHKLINE BEECHAM CORPORATION (US) 1997-07-10 WO disclosed