SCHEMBL8187488

SCHEMBL8187488

COc1cc(-c2c(C(F)(F)F)n[nH]c2-c2ccc(SCOC(C)=O)cc2)ccc1Br

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GRK6 P43250 4/20 0.33
HDAC3 O15379 1/20 0.33
HDAC4 P56524 1/20 0.33
HDAC1 Q13547 1/20 0.33
HDAC7 Q8WUI4 1/20 0.33
HDAC2 Q92769 1/20 0.33
HDAC10 Q969S8 1/20 0.33
HDAC11 Q96DB2 1/20 0.33
HDAC8 Q9BY41 1/20 0.33
HDAC6 Q9UBN7 1/20 0.33
HDAC9 Q9UKV0 1/20 0.33
HDAC5 Q9UQL6 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.32
TUBB4A P04350 1/20 0.32
TUBB P07437 1/20 0.32
TUBA3C P0DPH7 1/20 0.32
TUBA1B P68363 1/20 0.32
TUBA4A P68366 1/20 0.32
TUBB4B P68371 1/20 0.32
TUBB3 Q13509 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8188505 0.82 KDM4E (0.36) MAPTFYNCYP1A2KDM4EALDH1A1
SCHEMBL8187508 0.80 MEN1 (0.33) MEN1CYP1A2CYP2C9CYP2C19KMT2A
SCHEMBL8196758 0.80 MEN1 (0.33) MAPTMEN1CYP1A2CYP2C9CYP2C19
SCHEMBL8188363 0.77 FYN (0.38) MAPTFYNALDH1A1
SCHEMBL8199147 0.76 KMO (0.36) GRK6MAPTMEN1KMT2AHTT
SCHEMBL8201315 0.76 KDM4E (0.34) MAPTFYNKDM4EALDH1A1
SCHEMBL8195802 0.75 NR1H2 (0.37) MAPTFYNKMT2ASMN1; SMN2ALDH1A1
SCHEMBL8187466 0.71 PTGS2 (0.39) MEN1KMT2ASMN1; SMN2ALDH1A1
SCHEMBL8195825 0.70 PTGS2 (0.38) MEN1KMT2AHTTSMN1; SMN2ALDH1A1
SCHEMBL8200042 0.69 AR (0.37) ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed