SCHEMBL8199147

SCHEMBL8199147

COc1cc(-c2c(Cl)n[nH]c2-c2ccc(SCOC(C)=O)cc2)ccc1Cl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMO O15229 1/20 0.36
GRK6 P43250 3/20 0.35
HTT P42858 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MAPK10 P53779 1/20 0.35
RIPK2 O43353 1/20 0.34
ALDH1A1 P00352 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
DYRK1A Q13627 1/20 0.33
MAPT P10636 3/20 0.33
RET P07949 1/20 0.33
PTPN11 Q06124 1/20 0.33
POLB P06746 1/20 0.33
KDM4E B2RXH2 1/20 0.32
MEN1 O00255 1/20 0.32
GAA P10253 1/20 0.32
KMT2A Q03164 1/20 0.32
KDM5A P29375 1/20 0.32
KDM4C Q9H3R0 1/20 0.32
KDM5B Q9UGL1 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195495 0.84 TP53 (0.37) HTTSMN1; SMN2ALDH1A1NPSR1MAPT
SCHEMBL8195834 0.84 IKBKE (0.39) GRK6SMN1; SMN2ALDH1A1DYRK1AMAPT
SCHEMBL8200074 0.83 LMNA (0.38) HTTSMN1; SMN2MAPK10MAPTPOLB
SCHEMBL8195725 0.83 RPS6KA3 (0.40) GRK6HTTSMN1; SMN2MAPK10ALDH1A1
SCHEMBL8196103 0.83 GRK6 (0.38) GRK6SMN1; SMN2ALDH1A1MAPTMEN1
SCHEMBL8197299 0.82 MAPK14 (0.38) HTTSMN1; SMN2MAPK10ALDH1A1MAPT
SCHEMBL8196169 0.81 ALDH1A1 (0.37) KMOSMN1; SMN2RIPK2ALDH1A1MAPT
SCHEMBL8188126 0.73 MEN1 (0.40) HTTSMN1; SMN2ALDH1A1MEN1GAA
SCHEMBL8196014 0.72 ALDH1A1 (0.37) KMOSMN1; SMN2ALDH1A1MAPT
SCHEMBL8196005 0.72 MEN1 (0.39) HTTSMN1; SMN2ALDH1A1MEN1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed