SCHEMBL8196758

SCHEMBL8196758

CC(=O)OCSc1ccc(-c2[nH]nc(C(F)(F)F)c2-c2ccc(C(C)C)cc2)cc1

nearest known ligand 0.33

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 3/20 0.33
KMT2A Q03164 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CYP2C19 P33261 1/20 0.33
MAPT P10636 2/20 0.31
TP53 P04637 1/20 0.31
ALDH1A1 P00352 2/20 0.31
HTT P42858 2/20 0.31
LMNA P02545 1/20 0.31
HPGD P15428 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8187508 0.86 MEN1 (0.33) MEN1KMT2ASMN1; SMN2CYP1A2CYP2C9
SCHEMBL8197299 0.76 MAPK14 (0.38) MEN1KMT2ASMN1; SMN2CYP1A2MAPT
SCHEMBL8195495 0.76 TP53 (0.37) MEN1KMT2ASMN1; SMN2MAPTTP53
SCHEMBL8195725 0.75 RPS6KA3 (0.40) MEN1KMT2ASMN1; SMN2MAPTALDH1A1
SCHEMBL8200074 0.75 LMNA (0.38) MEN1KMT2ASMN1; SMN2MAPTTP53
SCHEMBL8197275 0.71 ALDH1A1 (0.36) SMN1; SMN2MAPTALDH1A1HTTLMNA
SCHEMBL8195827 0.70 PTGS2 (0.40) KMT2ACYP1A2CYP2C19TP53ALDH1A1
SCHEMBL8195834 0.69 IKBKE (0.39) SMN1; SMN2MAPTTP53ALDH1A1
SCHEMBL8196103 0.69 GRK6 (0.38) MEN1KMT2ASMN1; SMN2MAPTTP53
SCHEMBL8199147 0.68 KMO (0.36) MEN1KMT2ASMN1; SMN2MAPTALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO claimed
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed