Predicted protein targets (top 11)
| gene | UniProt | supporting neighbours | confidence | |
|---|---|---|---|---|
| ▸ | ELANE | P08246 | 1/20 | 0.37 |
| ▸ | ATM | Q13315 | 2/20 | 0.33 |
| ▸ | MAPT | P10636 | 2/20 | 0.33 |
| ▸ | PDE5A | O76074 | 1/20 | 0.33 |
| ▸ | TDP1 | Q9NUW8 | 1/20 | 0.33 |
| ▸ | PARP1 | P09874 | 1/20 | 0.32 |
| ▸ | HPSE | Q9Y251 | 1/20 | 0.32 |
| ▸ | KMT2A | Q03164 | 1/20 | 0.32 |
| ▸ | SLC22A6 | Q4U2R8 | 1/20 | 0.32 |
| ▸ | MAOB | P27338 | 1/20 | 0.30 |
| ▸ | ADORA2A | P29274 | 1/20 | 0.30 |
Click a target to see other patent compounds predicted against it — the reverse direction, in place.
Similar compounds — the chemically nearest patent molecules
Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.
| Compound | similarity | top predicted | shared targets | |
|---|---|---|---|---|
| SCHEMBL8844752 | 0.89 | MAPT (0.33) | ATMMAPTPDE5ATDP1PARP1 | |
| SCHEMBL27561443 | 0.88 | PDE5A (0.39) | ELANEATMPDE5ATDP1PARP1 | |
| SCHEMBL7707716 | 0.86 | SLC22A6 (0.44) | MAPTPDE5ATDP1KMT2ASLC22A6 | |
| SCHEMBL27464332 | 0.85 | ATM (0.34) | ATMMAPTTDP1PARP1HPSE | |
| SCHEMBL44289 | 0.83 | MAPT (0.33) | MAPTPARP1HPSEMAOBADORA2A | |
| SCHEMBL44290 | 0.81 | LMNA (0.35) | MAPTTDP1KMT2AMAOBADORA2A | |
| SCHEMBL5585189 | 0.80 | GABRG2 (0.35) | ELANEMAPTPDE5AKMT2AMAOB | |
| SCHEMBL14690221 | 0.80 | MAPT (0.32) | MAPTPARP1 | |
| SCHEMBL2534586 | 0.80 | MEN1 (0.38) | MAPTPARP1KMT2A | |
| SCHEMBL8590357 | 0.79 | THRB (0.38) | MAPTTDP1KMT2A |
Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.
Patent provenance — the patents this molecule appears in, and who filed them
Claimed or disclosed in 77 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.
| Patent | Title | Assignee | Published | Priority | Filing | Country | Status |
|---|---|---|---|---|---|---|---|
| US-20080031918-A1 | BARRIERS FOR POLYMERIC COATINGS | SURMODICS, INC. | 2008-02-07 | — | — | US | claimed |
| EP-1567203-B1 | BARRIERS FOR BIOACTIVE AGENT-CONTAINING POLYMERIC COATINGS | SURMODICS INC (US) | 2007-09-26 | — | — | EP | claimed |
| JP-3954616-B2 | — | — | 2007-08-08 | — | — | JP | claimed |
| US-7097850-B2 | Bioactive agent release coating and controlled humidity method | SURMODICS, INC. (US) | 2006-08-29 | — | — | US | claimed |
| EP-1551469-B1 | BIOACTIVE AGENT RELEASE COATING WITH AROMATIC POLY(METH)ACRYLATES | SURMODICS INC (US) | 2006-03-08 | — | — | EP | claimed |
| JP-2006505303-A | — | — | 2006-02-16 | — | — | JP | claimed |
| EP-1567203-A2 | BARRIERS FOR BIOACTIVE AGENT-CONTAINING POLYMERIC COATINGS | SurModics, Inc. (US) | 2005-08-31 | — | — | EP | claimed |
| EP-1551469-A1 | BIOACTIVE AGENT RELEASE COATING WITH AROMATIC POLY(METH)ACRYLATES | SurModics, Inc. (US) | 2005-07-13 | — | — | EP | claimed |
| EP-1534354-A1 | METHOD AND SYSTEM FOR PROVIDING BIOACTIVE AGENT RELEASE COATING | SurModics, Inc. (US) | 2005-06-01 | — | — | EP | claimed |
| EP-1517714-A1 | BIOACTIVE AGENT RELEASE COATING AND CONTROLLED HUMIDITY METHOD | SurModics, Inc. (US) | 2005-03-30 | — | — | EP | claimed |
| WO-2004052420-A2 | BARRIERS FOR BIOACTIVE AGENT-CONTAINING POLYMERIC COATINGS | SURMODICS, INC. (US) | 2004-06-24 | — | — | WO | claimed |
| US-20040111144-A1 | Barriers for polymeric coatings | Surmodics Coatings, LLC | 2004-06-10 | — | — | US | claimed |
| WO-2003105920-A1 | METHOD AND SYSTEM FOR PROVIDING BIOACTIVE AGENT RELEASE COATING | SURMODICS, INC. (US) | 2003-12-24 | — | — | WO | claimed |
| WO-2003105918-A1 | BIOACTIVE AGENT RELEASE COATING WITH AROMATIC POLY(METH)ACRYLATES | SURMODICS, INC. (US) | 2003-12-24 | — | — | WO | claimed |
| WO-2003105919-A1 | BIOACTIVE AGENT RELEASE COATING AND CONTROLLED HUMIDITY METHOD | SURMODICS, INC. (US) | 2003-12-24 | — | — | WO | claimed |
| US-20030232122-A1 | Bioactive agent release coating and controlled humidity method | Surmodics Coatings, LLC | 2003-12-18 | — | — | US | claimed |
| US-20030232087-A1 | Bioactive agent release coating with aromatic poly(meth)acrylates | Surmodics Coatings, LLC | 2003-12-18 | — | — | US | claimed |
| US-20020188037-A1 | Method and system for providing bioactive agent release coating | Surmodics Coatings, LLC | 2002-12-12 | — | — | US | claimed |
| JP-5295303-A | — | — | None | — | — | JP | disclosed |
| EP-0049860-A1 | Process for the preparation of reactive thyroid gland hormones T3 and T4 derivatives that are capable of coupling, and their use | Roche Diagnostics GmbH (DE) | 1982-04-21 | — | — | EP | disclosed |