SCHEMBL8188595

SCHEMBL8188595

O=C(O)C1C(c2ccccc2)=C1c1ccc(Cl)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 1/20 0.54
LMNA P02545 2/20 0.53
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
CTRC Q99895 1/20 0.45
CNR1 P21554 2/20 0.42
KDM4E B2RXH2 1/20 0.41
GAA P10253 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MGLL Q99685 2/20 0.41
VCP P55072 1/20 0.41
CYP1B1 Q16678 1/20 0.41
MAOB P27338 1/20 0.41
ADORA3 P0DMS8 1/20 0.41
SLC6A3 Q01959 1/20 0.41
ADAMTS5 Q9UNA0 1/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
MMP2 P08253 1/20 0.40
EDNRB P24530 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7823315 0.87 LMNA (0.67) LMNACES2CES1KDM4EGAA
SCHEMBL8190432 0.83 OPRK1 (0.49) LMNAVCPMAOBSLC6A3TSHR
Bicarbonate SCHEMBL27486769 0.78 CYP1A2 (0.79) CYP1A2LMNACES2CES1CTRC
SCHEMBL8179771 0.78 ALDH1A1 (0.51) CYP1A2LMNAKDM4EL3MBTL1TSHR
SCHEMBL14957913 0.72 TPMT (0.44) LMNASLC6A3
SCHEMBL4454036 0.72 CYP1A2 (1.00) CYP1A2LMNACTRCKDM4EGAA
SCHEMBL183912 0.72 CYP1A2 (1.00) CYP1A2LMNACTRCKDM4EGAA
SCHEMBL10874927 0.71 SRD5A2 (0.65) CYP1A2LMNACES2CES1CTRC
SCHEMBL9647503 0.71 CES2 (0.79) CYP1A2CES2CES1CTRCKDM4E
SCHEMBL2918529 0.71 LMNA (0.52) LMNAGAASLC6A3TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6020519-A Diphenyl-cyclopropenes as selective K-agonists WARNER-LAMBERT COMPANY (US) 2000-02-01 US claimed
WO-1998003491-A1 DIPHENYL-CYCLOPROPENES AS SELECTIVE K-AGONISTS WARNER-LAMBERT COMPANY (US) 1998-01-29 WO claimed
US-6020519-A Diphenyl-cyclopropenes as selective K-agonists WARNER-LAMBERT COMPANY (US) 2000-02-01 US disclosed
US-5968968-A Diphenyl-cyclopropenes as selective K-agonists WARNER-LAMBERT COMPANY (US) 1999-10-19 US disclosed
WO-1998003491-A1 DIPHENYL-CYCLOPROPENES AS SELECTIVE K-AGONISTS WARNER-LAMBERT COMPANY (US) 1998-01-29 WO disclosed