SCHEMBL8192539

SCHEMBL8192539

CCOC(=O)c1c(CO)c(NC(=O)OCc2ccccc2)cn1-n1cc(NC(=O)OC(C)(C)C)c(COC)c1C(=O)OCC

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
SYK P43405 1/20 0.41
CRHBP P24387 1/20 0.39
CRHR2 Q13324 1/20 0.39
BRD4 O60885 1/20 0.37
NAMPT P43490 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.36
KMT2A Q03164 1/20 0.35
P2RX7 Q99572 1/20 0.35
CTSS P25774 1/20 0.35
MKNK2 Q9HBH9 1/20 0.35
CNR2 P34972 1/20 0.35
TACR3 P29371 1/20 0.35
FAAH O00519 1/20 0.35
MGLL Q99685 1/20 0.35
BRD9 Q9H8M2 1/20 0.35
KDM4E B2RXH2 1/20 0.34
HSD17B10 Q99714 1/20 0.34
TOP2A P11388 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7669102 0.74 CRHBP (0.43) NPC1RAB9ASYKCRHBPCRHR2
SCHEMBL7660400 0.70 RAB9A (0.52) NPC1RAB9ANAMPTSMN1; SMN2KMT2A
SCHEMBL8184184 0.70 RAB9A (0.52) NPC1RAB9ANAMPTSMN1; SMN2KMT2A
SCHEMBL7661047 0.69 RAB9A (0.54) NPC1RAB9ACRHBPCRHR2NAMPT
SCHEMBL7043026 0.69 POLB (0.62) NPC1RAB9ASYKSMN1; SMN2KMT2A
SCHEMBL7661054 0.69 RAB9A (0.53) NPC1RAB9ANAMPTSMN1; SMN2KMT2A
SCHEMBL12872990 0.68 ALDH1A1 (0.56) NPC1RAB9ASYKSMN1; SMN2KMT2A
SCHEMBL31455060 0.68 NPC1 (0.55) NPC1RAB9ASYKSMN1; SMN2KMT2A
SCHEMBL28493853 0.68 KDM4E (0.60) SMN1; SMN2KMT2AKDM4EHSD17B10
SCHEMBL7400180 0.68 MGLL (0.50) NPC1RAB9ASYKSMN1; SMN2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0968186-A1 IMPROVED POLYAMIDES FOR BINDING IN THE MINOR GROOVE OF DOUBLE STRANDED DNA CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 2000-01-05 EP disclosed
WO-1998037066-A1 IMPROVED POLYAMIDES FOR BINDING IN THE MINOR GROOVE OF DOUBLE STRANDED DNA CALIFORNIA INSTITUTE OF TECHNOLOGY (US) 1998-08-27 WO disclosed