SCHEMBL8196142

SCHEMBL8196142

Cc1ccc(-c2c(Cl)n[nH]c2-c2ccc(S(=O)(=O)CCCO)cc2)cc1F

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
PTGS2 P35354 8/20 0.37
CA2 P00918 4/20 0.37
PTGDR2 Q9Y5Y4 1/20 0.37
PTGS1 P23219 3/20 0.35
BRD4 O60885 1/20 0.35
BRD2 P25440 1/20 0.35
BRD3 Q15059 1/20 0.35
NR1H2 P55055 1/20 0.34
NR1H3 Q13133 1/20 0.34
ALDH1A1 P00352 1/20 0.33
MAPT P10636 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8188503 0.92 PTGS2 (0.40) PTGS2CA2PTGDR2PTGS1NR1H2
SCHEMBL8200031 0.90 PTGS2 (0.39) PTGS2CA2PTGDR2PTGS1BRD4
SCHEMBL8196899 0.88 PTGS2 (0.39) PTGS2CA2PTGDR2PTGS1BRD4
SCHEMBL8195877 0.85 PTGS2 (0.41) PTGS2CA2PTGDR2PTGS1ALDH1A1
SCHEMBL8196926 0.85 CA2 (0.42) PTGS2CA2PTGS1ALDH1A1
SCHEMBL8196062 0.85 ALDH1A1 (0.46) PTGS2CA2ALDH1A1MAPT
SCHEMBL8199737 0.83 PTGS2 (0.40) PTGS2CA2PTGDR2PTGS1BRD4
SCHEMBL8202075 0.83 PTGS2 (0.37) PTGS2PTGS1MAPT
SCHEMBL8068397 0.82 PTGS2 (0.53) PTGS2
SCHEMBL8196010 0.82 CA2 (0.43) PTGS2CA2PTGDR2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed