SCHEMBL8197299

SCHEMBL8197299

CC(=O)OCSc1ccc(-c2[nH]nc(Cl)c2-c2ccc(F)cc2)cc1

nearest known ligand 0.38

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MAPK14 Q16539 4/20 0.38
MAPT P10636 3/20 0.35
TP53 P04637 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.34
TDP1 Q9NUW8 1/20 0.32
RAB9A P51151 1/20 0.32
POLB P06746 1/20 0.32
RXFP1 Q9HBX9 1/20 0.32
CYP1A2 P05177 1/20 0.32
GSK3B P49841 1/20 0.32
KMT2A Q03164 3/20 0.32
NPC1 O15118 1/20 0.32
HTT P42858 2/20 0.31
MAPK10 P53779 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MEN1 O00255 2/20 0.31
ALDH1A1 P00352 2/20 0.31
PTGS2 P35354 1/20 0.31
ILK Q13418 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195495 0.91 TP53 (0.37) MAPK14MAPTTP53RAB9AKMT2A
SCHEMBL8200074 0.90 LMNA (0.38) MAPTTP53L3MBTL1POLBGSK3B
SCHEMBL8195725 0.90 RPS6KA3 (0.40) MAPK14MAPTL3MBTL1RAB9AKMT2A
SCHEMBL8195834 0.84 IKBKE (0.39) MAPTTP53GSK3BSMN1; SMN2ALDH1A1
SCHEMBL8196103 0.83 GRK6 (0.38) MAPTTP53L3MBTL1KMT2ASMN1; SMN2
SCHEMBL8199147 0.82 KMO (0.36) MAPTPOLBKMT2AHTTMAPK10
SCHEMBL8639382 0.77 MAPK14 (0.44) MAPK14GSK3BPTGS2
SCHEMBL8187508 0.74 MEN1 (0.33) CYP1A2KMT2ASMN1; SMN2MEN1
SCHEMBL6180868 0.72 PTGS2 (0.55) MAPK14PTGS2
SCHEMBL8202075 0.68 PTGS2 (0.37) MAPTKMT2AHTTMEN1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed