SCHEMBL8199643

SCHEMBL8199643

COC(=O)c1cccc2c1CCC(CCN1CCC(c3ccccc3)CC1)C2=O

nearest known ligand 0.48

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
CCR5 P51681 1/20 0.48
SLC18A3 Q16572 2/20 0.47
HTR2C P28335 3/20 0.46
HTR7 P34969 3/20 0.44
SIGMAR1 Q99720 2/20 0.43
CARM1 Q86X55 1/20 0.43
PRMT6 Q96LA8 1/20 0.43
PRCP P42785 2/20 0.43
DRD2 P14416 1/20 0.43
DRD3 P35462 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200402 0.89 HTR2C (0.48) CCR5SLC18A3HTR2CHTR7SIGMAR1
Hydrochloric Acid SCHEMBL8199293 0.86 HTR2C (0.46) SLC18A3HTR2CHTR7SIGMAR1PRCP
SCHEMBL8203549 0.84 HTR2C (0.43) HTR2CHTR7DRD2DRD3
SCHEMBL8203504 0.83 HTR2C (0.42) SLC18A3HTR2CHTR7SIGMAR1CARM1
SCHEMBL8198484 0.83 HTR2C (0.42) SLC18A3HTR2CHTR7SIGMAR1CARM1
SCHEMBL8200968 0.83 CCR5 (0.44) CCR5SLC18A3HTR2CHTR7SIGMAR1
SCHEMBL8192538 0.83 PRCP (0.56) CCR5SLC18A3HTR2CPRCP
SCHEMBL8199832 0.83 PRCP (0.56) CCR5SLC18A3HTR2CPRCP
SCHEMBL8203121 0.82 DRD3 (0.43) SLC18A3HTR2CCARM1PRMT6DRD2
SCHEMBL8203423 0.82 DRD3 (0.43) SLC18A3HTR2CHTR7SIGMAR1CARM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO disclosed