SCHEMBL8192538

SCHEMBL8192538

C[C@@H](NC(=O)c1cccc2c1CCC(CCN1CCC(c3ccccc3)CC1)C2=O)c1ccccc1

nearest known ligand 0.56

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PRCP P42785 7/20 0.56
HTR2C P28335 1/20 0.41
SLC18A3 Q16572 1/20 0.40
ITGA4 P13612 1/20 0.40
ITGB7 P26010 1/20 0.40
ADRA1D P25100 1/20 0.40
ADRA1A P35348 1/20 0.40
ADRA1B P35368 1/20 0.40
CCR5 P51681 1/20 0.40
KDM4E B2RXH2 1/20 0.39
ALDH1A1 P00352 1/20 0.39
LMNA P02545 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
PPARG P37231 1/20 0.39
MAPK1 P28482 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199832 1.00 PRCP (0.56) PRCPHTR2CSLC18A3ITGA4ITGB7
SCHEMBL8200402 0.84 HTR2C (0.48) PRCPHTR2CSLC18A3CCR5
SCHEMBL8199643 0.83 CCR5 (0.48) PRCPHTR2CSLC18A3CCR5
SCHEMBL8198484 0.83 HTR2C (0.42) HTR2CSLC18A3
SCHEMBL8203423 0.81 DRD3 (0.43) PRCPHTR2CSLC18A3ADRA1DADRA1A
SCHEMBL8203121 0.81 DRD3 (0.43) HTR2CSLC18A3ADRA1DADRA1AADRA1B
SCHEMBL8200414 0.81 PRCP (0.44) PRCPHTR2CSLC18A3CCR5ALDH1A1
SCHEMBL8589678 0.81 SIGMAR1 (0.44) HTR2CKDM4E
SCHEMBL8588349 0.81 SIGMAR1 (0.44) HTR2CKDM4E
SCHEMBL8200419 0.81 SIGMAR1 (0.44) HTR2CKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed